SCHEMBL9562378

SCHEMBL9562378

CCCC(=O)Oc1ccc(OC(=O)c2ccc(OCC)cc2)c(F)c1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
CCNC P24863 1/20 0.47
CDK8 P49336 1/20 0.47
NPC1 O15118 1/20 0.47
MAPT P10636 3/20 0.46
THRB P10828 1/20 0.46
PARP10 Q53GL7 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HPGD P15428 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GAA P10253 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
ALOX15 P16050 1/20 0.44
PLK1 P53350 1/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
SCN1A P35498 1/20 0.43
SCN2A Q99250 1/20 0.43
SCN3A Q9NY46 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9475988 0.84 NPC1 (0.54) KMT2ANPC1MAPTTHRBLMNA
SCHEMBL10418697 0.80 BCL9 (0.40) KMT2ANPC1MAPTTHRBHPGD
SCHEMBL9406188 0.80 PRSS1 (0.47) KMT2ACCNCCDK8NPC1MAPT
SCHEMBL1994064 0.79 ALOX15 (0.49) KMT2AALOX15ALDH1A1LMNAMEN1
SCHEMBL14766407 0.79 MAPT (0.48) KMT2ACCNCCDK8NPC1MAPT
SCHEMBL14767194 0.79 MAPT (0.48) KMT2ACCNCCDK8NPC1MAPT
SCHEMBL10418081 0.79 KMT2A (0.46) KMT2ACCNCCDK8NPC1MAPT
SCHEMBL20703605 0.77 BCL9 (0.60) KMT2ANPC1MAPTPARP10L3MBTL1
SCHEMBL9405801 0.77 NPC1 (0.59) KMT2ANPC1MAPTLMNA
SCHEMBL10381844 0.77 MAPT (0.47) KMT2ANPC1MAPTTHRBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5248447-A 2,3-difluorohydroquinone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-09-28 US disclosed
EP-0518961-A1 DERIVATIVES OF GLYCINAMIDE, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Aventis Pharma S.A. (FR) 1992-12-23 EP disclosed