SCHEMBL9562884

SCHEMBL9562884

CCCC[Sn](C=Cc1c(-c2ccc(F)cc2)nc(-c2ccccc2)nc1C(C)C)(CCCC)CCCC

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 7/20 0.54
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
PDE6D O43924 1/20 0.40
NR1I2 O75469 1/20 0.40
PDE4D Q08499 1/20 0.40
DPP4 P27487 1/20 0.39
GCGR P47871 4/20 0.36
ABCC3 O15438 1/20 0.35
ABCC4 O15439 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9562755 0.79 HMGCR (0.56) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL9562749 0.79 HMGCR (0.56) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL9521683 0.79 HMGCR (0.53) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10433924 0.77 HMGCR (0.57) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10434205 0.77 HMGCR (0.57) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL8846369 0.77 HMGCR (0.53) HMGCRALDH1A1CYP3A4DPP4GCGR
SCHEMBL9562922 0.77 HMGCR (0.56) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10433897 0.75 HMGCR (0.55) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL10433896 0.75 HMGCR (0.55) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL8952918 0.75 HMGCR (0.43) HMGCRGCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202327-A PHOSPHORUS-CONTAINING HMG-COA REDUCTASE INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1993-04-13 US disclosed
EP-0522431-A1 Phophorus-containing HMG-COA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1993-01-13 EP disclosed