SCHEMBL9563279

SCHEMBL9563279

CC(CCN1CCC(OC(c2ccccc2)c2cccs2)CC1)Oc1ccccc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 5/20 0.42
CYP2D6 P10635 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP2C19 P33261 1/20 0.40
SLC6A2 P23975 3/20 0.38
OPRM1 P35372 2/20 0.38
CHRM2 P08172 2/20 0.38
HTR1A P08908 2/20 0.38
ADRA2A P08913 2/20 0.38
CHRM1 P11229 2/20 0.38
DRD1 P21728 2/20 0.38
ADRA1A P35348 2/20 0.38
DRD3 P35462 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNH2 Q12809 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
OPRL1 P41146 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A4 P31645 2/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9563288 0.90 BCHE (0.49) BCHECYP2D6KDM4ECYP2C19SLC6A2
SCHEMBL9563207 0.85 CYP2D6 (0.52) BCHECYP2D6KDM4ECYP2C19NPC1
SCHEMBL9563318 0.85 HTR1A (0.41) BCHECYP2D6SLC6A2OPRM1CHRM2
Hydrochloric Acid SCHEMBL9563227 0.84 CYP2D6 (0.52) BCHECYP2D6KDM4ECYP2C19
SCHEMBL9563187 0.82 CCR5 (0.38) BCHECYP2D6SLC6A2OPRM1CHRM2
SCHEMBL9563257 0.81 CYP2D6 (0.40) BCHECYP2D6KDM4ECYP2C19SLC6A2
SCHEMBL9565888 0.80 BCHE (0.38) BCHECYP2D6KDM4ECYP2C19SLC6A3
SCHEMBL9563330 0.80 BCHE (0.38) BCHECYP2D6KDM4ECYP2C19SLC6A3
SCHEMBL9563326 0.80 BCHE (0.38) BCHECYP2D6KDM4ECYP2C19SLC6A3
SCHEMBL9563202 0.79 CYP2D6 (0.55) BCHECYP2D6KDM4ECYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529365-A1 Diarylmethoxypiperidine derivatives Kaken Pharmaceutical Co., Ltd. (JP) 1993-03-03 EP disclosed
US-5190959-A Antihistamines, antiallergens, treatment of ischemic heart disease KAKEN PHARMACEUTICAL CO. LTD. (JP) 1993-03-02 US disclosed