SCHEMBL9563286

SCHEMBL9563286

O=[N+]([O-])c1ccccc1OCCCN1CCC(O)CC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.70
CYP2C19 P33261 2/20 0.70
CYP1A2 P05177 1/20 0.70
KDM4E B2RXH2 6/20 0.69
ALDH1A1 P00352 6/20 0.60
SMN1; SMN2 Q16637 4/20 0.59
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
RECQL P46063 1/20 0.56
TDP1 Q9NUW8 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
LTA4H P09960 1/20 0.51
PTGS1 P23219 1/20 0.51
PTGS2 P35354 1/20 0.51
SIGMAR1 Q99720 2/20 0.50
PKM P14618 1/20 0.49
STAT1 P42224 1/20 0.49
HTT P42858 1/20 0.49
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9563362 0.96 CYP2D6 (0.74) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563282 0.95 CYP2D6 (0.72) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563345 0.94 KDM4E (0.64) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563233 0.86 ALDH1A1 (0.53) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563198 0.83 ALDH1A1 (0.71) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563181 0.83 ALDH1A1 (0.69) CYP2D6CYP2C19KDM4EALDH1A1SMN1; SMN2
SCHEMBL9563398 0.81 KDM4E (0.50) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563333 0.81 CYP2D6 (0.60) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563281 0.80 RAB9A (0.51) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1
SCHEMBL9563172 0.80 RAB9A (0.51) CYP2D6CYP2C19CYP1A2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529365-A1 Diarylmethoxypiperidine derivatives Kaken Pharmaceutical Co., Ltd. (JP) 1993-03-03 EP disclosed
US-5190959-A Antihistamines, antiallergens, treatment of ischemic heart disease KAKEN PHARMACEUTICAL CO. LTD. (JP) 1993-03-02 US disclosed