SCHEMBL9564189

SCHEMBL9564189

COC(=O)c1ccc(Cc2c[nH]c3nc(N)nc(O)c23)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.41
NPC1 O15118 1/20 0.40
MPO P05164 1/20 0.38
DPP4 P27487 2/20 0.37
TYMS P04818 5/20 0.36
CDC7 O00311 1/20 0.36
NTRK1 P04629 1/20 0.36
DHFR P00374 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4215783 0.79 TLR7 (0.47) MPODPP4DHFRCYP1A2CYP3A4
SCHEMBL14329878 0.78 DHFR (0.51) NPC1TYMSDHFRCYP1A2CYP3A4
SCHEMBL9564217 0.78 L3MBTL1 (0.45) TYMSDHFR
SCHEMBL9564219 0.78 L3MBTL1 (0.45) TYMSDHFR
SCHEMBL9564240 0.78 DHFR (0.58) TYMSDHFR
Guanidine SCHEMBL2854796 0.74 TLR7 (0.43) MPODPP4DHFR
SCHEMBL9564205 0.74 TYMS (0.43) TYMSDHFR
SCHEMBL2852426 0.73 NPSR1 (0.48) DPP4DHFR
SCHEMBL9564224 0.70 MAPT (0.37) NPC1TYMSDHFRCYP3A4
SCHEMBL9044792 0.69 TYMS (0.51) NPC1TYMSDHFRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed