SCHEMBL9564816

SCHEMBL9564816

CCOC(=O)N1CCC(Nc2nc3cncnc3n2Cc2ccco2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 5/20 0.46
ALDH1A1 P00352 6/20 0.45
HSD17B10 Q99714 3/20 0.45
KDM4E B2RXH2 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NOS1 P29475 4/20 0.44
NOS3 P29474 2/20 0.44
HPGD P15428 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MAP4K4 O95819 1/20 0.43
ADORA3 P0DMS8 4/20 0.42
ADORA2A P29274 4/20 0.42
ADORA1 P30542 4/20 0.42
ADORA2B P29275 2/20 0.42
TSHR P16473 3/20 0.42
MAPT P10636 2/20 0.42
MAPK1 P28482 1/20 0.42
ATM Q13315 1/20 0.42
CDK1 P06493 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9385081 0.88 NOS2 (0.52) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL10875714 0.87 ALDH1A1 (0.38) ALDH1A1HSD17B10KDM4ESMN1; SMN2HPGD
SCHEMBL9564774 0.87 ALDH1A1 (0.44) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL9564864 0.86 ALDH1A1 (0.51) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL9630462 0.85 NOS2 (0.48) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL9564849 0.85 SMN1; SMN2 (0.50) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL9602879 0.84 NOS2 (0.56) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL7492660 0.84 ALDH1A1 (0.53) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL9629563 0.83 NOS2 (0.46) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2
SCHEMBL9564902 0.83 USP2 (0.51) NOS2ALDH1A1HSD17B10KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed