SCHEMBL9564879

SCHEMBL9564879

Cc1nc2ccccn2c(=O)c1CCN1CCC(S(=O)(=O)c2nc3cncnc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 13/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
TSHR P16473 4/20 0.53
CYP2D6 P10635 3/20 0.53
HPGD P15428 2/20 0.53
HTR1A P08908 2/20 0.53
HTR2C P28335 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
MAPT P10636 1/20 0.53
PKM P14618 1/20 0.53
THPO P40225 1/20 0.53
PMP22 Q01453 1/20 0.53
KMT2A Q03164 1/20 0.53
ACHE P22303 1/20 0.49
CYP1A2 P05177 14/20 0.47
USP2 O75604 12/20 0.47
CYP2C9 P11712 11/20 0.47
CYP2C19 P33261 10/20 0.47
HIF1A Q16665 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564945 0.85 CYP3A4 (0.54) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
SCHEMBL9691198 0.83 CYP3A4 (0.51) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
Fumaric Acid SCHEMBL9807342 0.79 CYP3A4 (0.50) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
SCHEMBL9537351 0.76 HTR1A (0.56) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
Hydrochloric Acid SCHEMBL9800689 0.75 HTR1A (0.54) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
Fumaric Acid SCHEMBL9876528 0.74 HRH1 (0.49) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
SCHEMBL9536711 0.74 CYP2D6 (0.59) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
SCHEMBL9564962 0.73 USP2 (0.50) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
SCHEMBL9564997 0.73 CYP3A4 (0.47) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD
SCHEMBL9564953 0.73 CYP1A2 (0.54) CYP3A4SMN1; SMN2TSHRCYP2D6HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed