SCHEMBL9564906

SCHEMBL9564906

c1ccc(CCN2CCC(Nc3nc4cncnc4n3Cc3ccco3)CC2)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 2/20 0.39
KCNH2 Q12809 10/20 0.38
NR4A2 P43354 1/20 0.37
CYP1A2 P05177 3/20 0.36
CYP2D6 P10635 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
LMNA P02545 2/20 0.36
CYP3A4 P08684 2/20 0.36
MAPT P10636 2/20 0.36
CYP2C19 P33261 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HTR2A P28223 3/20 0.36
HRH1 P35367 2/20 0.36
MLNR O43193 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564838 0.90 SSTR5 (0.43) SSTR5KCNH2NR4A2CYP1A2CYP2D6
SCHEMBL9564808 0.87 HTR2A (0.38) SSTR5KCNH2NR4A2CYP1A2CYP2D6
SCHEMBL9565012 0.85 SSTR5 (0.39) SSTR5KCNH2NR4A2CYP1A2CYP2D6
SCHEMBL9564929 0.84 SSTR5 (0.57) SSTR5KCNH2NR4A2CYP1A2CYP2D6
SCHEMBL9564789 0.80 NR4A2 (0.42) KCNH2NR4A2CYP1A2CYP2D6MEN1
SCHEMBL9565084 0.79 KCNH2 (0.36) SSTR5KCNH2MEN1KMT2AMAPT
SCHEMBL9565053 0.79 KCNH2 (0.57) SSTR5KCNH2NR4A2CYP1A2CYP2D6
Water SCHEMBL9564806 0.79 NR4A2 (0.42) KCNH2NR4A2CYP1A2CYP2D6MEN1
Water SCHEMBL9564807 0.79 NR4A2 (0.42) KCNH2NR4A2CYP1A2CYP2D6MEN1
Hydrochloric Acid SCHEMBL9564793 0.77 ADRA1D (0.41) MAPTALDH1A1USP2HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed