SCHEMBL9566841

SCHEMBL9566841

CCCCc1ccc(NC(=O)c2ccc(CO)nc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 11/20 0.60
KDM4E B2RXH2 2/20 0.57
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
ALDH1A1 P00352 1/20 0.56
NFKB1 P19838 1/20 0.56
NFKB2 Q00653 1/20 0.56
RELA Q04206 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
GALR3 O60755 1/20 0.53
TP53 P04637 1/20 0.49
GAA P10253 1/20 0.49
POLB P06746 1/20 0.49
PLK1 P53350 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566731 0.87 TRPV1 (0.56) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL9566817 0.86 TRPV1 (0.55) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL13210620 0.86 NPC1 (0.67) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL9566843 0.85 TRPV1 (0.54) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL9566854 0.84 TRPV1 (0.53) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL9566764 0.82 TRPV1 (0.60) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL9566790 0.82 LMNA (0.59) KDM4ENPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL13989044 0.81 TRPV1 (0.59) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL9566836 0.81 TRPV1 (0.59) TRPV1KDM4ENPC1RAB9AALDH1A1
SCHEMBL9566887 0.80 P4HTM (0.69) KDM4ENPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533130-A1 2-Hydroxymethylpyridines, the corresponding pyridine-N-oxides and derivatives thereof, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-24 EP disclosed