SCHEMBL9566883

SCHEMBL9566883

CC(=O)OCc1ccc(C(=O)Nc2ccc(Oc3ccc(F)cc3)cc2)cn1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 13/20 0.52
CXCR1 P25024 11/20 0.52
P4HTM Q9NXG6 2/20 0.50
F2 P00734 1/20 0.47
PLG P00747 1/20 0.47
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
ST14 Q9Y5Y6 1/20 0.47
ALDH1A1 P00352 1/20 0.47
BRAF P15056 1/20 0.47
HDAC1 Q13547 1/20 0.47
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566786 0.94 CXCR2 (0.57) CXCR2CXCR1P4HTMALDH1A1
SCHEMBL9566811 0.89 CXCR2 (0.57) CXCR2CXCR1P4HTMF2PLG
SCHEMBL9566753 0.87 CXCR2 (0.54) CXCR2CXCR1P4HTMF2PLG
SCHEMBL9566799 0.86 CXCR2 (0.53) CXCR2CXCR1P4HTMMEN1LMNA
SCHEMBL9566849 0.85 P4HTM (0.63) P4HTMALDH1A1MEN1LMNAKMT2A
SCHEMBL9566852 0.85 P4HTM (0.55) CXCR2CXCR1P4HTMF2PLG
SCHEMBL9566814 0.83 P4HTM (0.47) CXCR2P4HTMMEN1LMNAKMT2A
SCHEMBL9566759 0.83 CXCR2 (0.55) CXCR2CXCR1P4HTMALDH1A1
SCHEMBL9566792 0.82 P4HTM (0.55) P4HTMALDH1A1MEN1LMNAKMT2A
SCHEMBL9566758 0.82 NPC1 (0.57) CXCR2CXCR1P4HTMALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533130-A1 2-Hydroxymethylpyridines, the corresponding pyridine-N-oxides and derivatives thereof, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-24 EP disclosed