SCHEMBL9566852

SCHEMBL9566852

O=C(Nc1ccc(Oc2ccc(F)cc2)cc1)c1ccc(CO)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 1/20 0.55
CXCR2 P25025 10/20 0.54
CXCR1 P25024 8/20 0.54
F2 P00734 1/20 0.52
PLG P00747 1/20 0.52
PRSS1 P07477 1/20 0.52
PRSS2 P07478 1/20 0.52
PRSS3 P35030 1/20 0.52
ST14 Q9Y5Y6 1/20 0.52
F13A1 P00488 1/20 0.49
TGM2 P21980 1/20 0.49
PTPN1 P18031 1/20 0.49
PTPN6 P29350 1/20 0.49
PTPN11 Q06124 1/20 0.49
ALDH1A1 P00352 1/20 0.48
BRAF P15056 1/20 0.48
HDAC1 Q13547 1/20 0.48
KMT2A Q03164 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566833 0.92 P4HTM (0.63) P4HTMCXCR2CXCR1PTPN1PTPN6
SCHEMBL9566811 0.87 CXCR2 (0.57) P4HTMCXCR2CXCR1F2PLG
SCHEMBL9566753 0.85 CXCR2 (0.54) P4HTMCXCR2CXCR1F2PLG
SCHEMBL9566883 0.85 CXCR2 (0.52) P4HTMCXCR2CXCR1F2PLG
SCHEMBL9566803 0.83 P4HTM (0.66) P4HTMALDH1A1KMT2ACYP1A2CYP3A4
SCHEMBL9566799 0.82 CXCR2 (0.53) P4HTMCXCR2CXCR1KMT2AKCNQ3
SCHEMBL9566829 0.82 CXCR2 (0.58) P4HTMCXCR2CXCR1HDAC1KMT2A
SCHEMBL9566887 0.82 P4HTM (0.69) P4HTMALDH1A1KMT2ACYP1A2CYP3A4
SCHEMBL9517015 0.82 P4HTM (0.51) P4HTMCXCR2CXCR1PTPN1PTPN6
SCHEMBL9566862 0.81 ABL1 (0.51) P4HTMKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533130-A1 2-Hydroxymethylpyridines, the corresponding pyridine-N-oxides and derivatives thereof, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-24 EP disclosed