SCHEMBL9566902

SCHEMBL9566902

COCc1ccc(C(=O)Nc2ccc(F)cc2)cn1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 15/20 0.62
CXCR1 P25024 12/20 0.62
P4HTM Q9NXG6 1/20 0.58
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
ATM Q13315 1/20 0.56
ALDH1A1 P00352 1/20 0.53
PTPN1 P18031 1/20 0.51
PTPN6 P29350 1/20 0.51
PTPN11 Q06124 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566811 0.94 CXCR2 (0.57) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9515480 0.90 CXCR2 (0.52) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9566786 0.87 CXCR2 (0.57) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9566868 0.87 CXCR2 (0.60) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9566851 0.87 P4HTM (0.58) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9566760 0.86 RAB9A (0.60) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9566759 0.85 CXCR2 (0.55) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9566791 0.85 P4HTM (0.62) CXCR2CXCR1P4HTMNPC1RAB9A
SCHEMBL9566897 0.85 P4HTM (0.66) P4HTMNPC1RAB9AALDH1A1
SCHEMBL12020864 0.84 MEN1 (0.70) CXCR2CXCR1P4HTMNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533130-A1 2-Hydroxymethylpyridines, the corresponding pyridine-N-oxides and derivatives thereof, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-24 EP disclosed