SCHEMBL9515480

SCHEMBL9515480

COCc1ccc(C(=O)NC(=O)Nc2ccc(F)cc2)cn1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 13/20 0.52
CXCR1 P25024 11/20 0.52
MEN1 O00255 2/20 0.49
MAPT P10636 2/20 0.49
KMT2A Q03164 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
MAPK1 P28482 1/20 0.49
HTT P42858 1/20 0.49
P4HTM Q9NXG6 1/20 0.47
CASP3 P42574 1/20 0.45
TRPV1 Q8NER1 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
ATM Q13315 1/20 0.45
ALDH1A1 P00352 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566902 0.90 CXCR2 (0.62) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL9519474 0.88 CXCR2 (0.50) CXCR2CXCR1MEN1MAPTKMT2A
SCHEMBL9516951 0.88 NPC1 (0.52) CXCR2CXCR1MEN1MAPTKMT2A
SCHEMBL9517015 0.85 P4HTM (0.51) CXCR2CXCR1MEN1MAPTKMT2A
SCHEMBL9566811 0.85 CXCR2 (0.57) CXCR2CXCR1MEN1KMT2ANPC1
SCHEMBL9519589 0.83 CXCR2 (0.54) CXCR2CXCR1MEN1KMT2AP4HTM
SCHEMBL9519137 0.78 NPC1 (0.54) MEN1MAPTKMT2ANPC1RAB9A
SCHEMBL9566868 0.78 CXCR2 (0.60) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL9566786 0.78 CXCR2 (0.57) CXCR2CXCR1NPC1RAB9AP4HTM
SCHEMBL3950709 0.78 BAZ2B (0.49) MEN1MAPTKMT2AHTTP4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1079466-A 4-or 5-(sulphur) acylimino-and (inferior sulphur) amidopyridine and pyridine-N-oxide thereof HOECHST AG (DE) 1993-12-15 CN disclosed
EP-0567997-A1 4- or 5-(sulf)imido- and (sulfon)amidopyridines and their pyridine-N-oxides, process for their preparation and their use as pharmaceutical HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-03 EP disclosed