SCHEMBL9567637

SCHEMBL9567637

CO[C@@H]1[C@@H](Cn2ccnc2)[C@H](CCc2cccc3ccccc23)CCC1(C)C

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
SLC18A2 Q05940 1/20 0.38
CYP19A1 P11511 3/20 0.35
TBXAS1 P24557 2/20 0.35
IDO1 P14902 1/20 0.35
FNTA P49354 5/20 0.34
FNTB P49356 5/20 0.34
PGGT1B P53609 2/20 0.34
CYP11B1 P15538 3/20 0.34
CYP11B2 P19099 3/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CYP17A1 P05093 1/20 0.32
QPCT Q16769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9244403 0.86 POLB (0.45) POLBSLC18A2CYP19A1TBXAS1IDO1
SCHEMBL9247259 0.84 POLB (0.47) POLBCYP19A1TBXAS1IDO1FNTA
SCHEMBL9247262 0.84 POLB (0.47) POLBCYP19A1TBXAS1IDO1FNTA
SCHEMBL9241703 0.84 CYP19A1 (0.47) POLBCYP19A1TBXAS1IDO1FNTA
SCHEMBL9567750 0.84 GAA (0.38) POLBSLC18A2SLC6A2SLC6A4
SCHEMBL9247365 0.80 SLC18A2 (0.42) SLC18A2SLC6A2SLC6A4
SCHEMBL8714592 0.76 TBXAS1 (0.40) CYP19A1TBXAS1
SCHEMBL9244400 0.71 CYP19A1 (0.45) POLBCYP19A1TBXAS1IDO1FNTA
SCHEMBL9243685 0.71 CALCA (0.35) CYP19A1CYP11B1CYP17A1
SCHEMBL9244604 0.70 CALCA (0.36) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0524439-A1 Novel cyclohexane and tetrahydropyran derivatives and antifungal compositions containing these derivatives F.HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT (CH) 1993-01-27 EP disclosed