SCHEMBL9568147

SCHEMBL9568147

COc1ccc(-c2ccc(C(=N)NC(=O)OCc3ccccc3)cc2)cc1C(=O)N[C@H]1CC[C@H](C(=O)OCOC(=O)C(C)(C)C)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.40
MCHR1 Q99705 1/20 0.39
CNR1 P21554 3/20 0.37
CNR2 P34972 3/20 0.37
ACHE P22303 3/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
LMNA P02545 1/20 0.36
EPHX1 P07099 1/20 0.36
CYP3A4 P08684 2/20 0.36
REN P00797 1/20 0.36
SMPD3 Q9NY59 1/20 0.35
DRD4 P21917 6/20 0.35
DRD3 P35462 3/20 0.35
NR1H4 Q96RI1 1/20 0.35
DRD2 P14416 2/20 0.35
CYP1A2 P05177 1/20 0.35
ADRA2A P08913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568142 1.00 ALDH1A1 (0.41) ALDH1A1GAATSHRMCHR1CNR1
SCHEMBL9568079 0.87 TSHR (0.43) ALDH1A1GAATSHRMCHR1CNR1
SCHEMBL9568082 0.86 TSHR (0.40) ALDH1A1GAATSHRMCHR1CNR1
SCHEMBL9568220 0.84 ST14 (0.40)
SCHEMBL9568223 0.84 ST14 (0.40)
SCHEMBL9568227 0.84 MCHR1 (0.40) ALDH1A1GAATSHRMCHR1CNR1
SCHEMBL9568230 0.84 MCHR1 (0.40) ALDH1A1GAATSHRMCHR1CNR1
SCHEMBL9568102 0.83 TSHR (0.39) ALDH1A1GAATSHRMCHR1CNR1
SCHEMBL9568097 0.83 TSHR (0.39) ALDH1A1GAATSHRMCHR1CNR1
SCHEMBL9568178 0.83 MCHR1 (0.39) ALDH1A1GAATSHRMCHR1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574808-A1 Amidine-biphenyl derivatives, process for their production & medical preparation containing them Dr. Karl Thomae GmbH (DE) 1993-12-22 EP disclosed