SCHEMBL9568178

SCHEMBL9568178

COc1ccc(-c2ccc(C(=N)NC(=O)OCc3ccccc3)cc2)cc1C(=O)N[C@H]1CC[C@H](C(=O)OCC(=O)N2CCOCC2)CC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.39
ALDH1A1 P00352 5/20 0.39
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
HPGD P15428 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KMT2A Q03164 1/20 0.38
TSHR P16473 1/20 0.37
USP2 O75604 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568177 1.00 MCHR1 (0.39) MCHR1ALDH1A1GAAKDM4EGLA
SCHEMBL9568230 0.93 MCHR1 (0.40) MCHR1ALDH1A1GAAKMT2ATSHR
SCHEMBL9568227 0.93 MCHR1 (0.40) MCHR1ALDH1A1GAAKMT2ATSHR
SCHEMBL9568082 0.86 TSHR (0.40) MCHR1ALDH1A1GAAKMT2ATSHR
Hydrochloric Acid SCHEMBL9568148 0.84 KMT2A (0.43) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL9568147 0.83 ALDH1A1 (0.41) MCHR1ALDH1A1GAATSHRDRD4
SCHEMBL9568142 0.83 ALDH1A1 (0.41) MCHR1ALDH1A1GAATSHRDRD4
SCHEMBL9568079 0.81 TSHR (0.43) MCHR1ALDH1A1GAATSHRDRD4
SCHEMBL9174514 0.80 HPGDS (0.42) ALDH1A1GAAKMT2ATSHRMAPT
SCHEMBL9568102 0.80 TSHR (0.39) MCHR1ALDH1A1GAATSHRDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574808-A1 Amidine-biphenyl derivatives, process for their production & medical preparation containing them Dr. Karl Thomae GmbH (DE) 1993-12-22 EP disclosed