SCHEMBL9568227

SCHEMBL9568227

COc1ccc(-c2ccc(C(=N)NC(=O)OCc3ccccc3)cc2)cc1C(=O)NC1CCC(C(=O)OCC(=O)N2CCCCC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.40
KCNH2 Q12809 2/20 0.40
DPP4 P27487 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
TSHR P16473 1/20 0.38
EPHX1 P07099 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
ALDH1A1 P00352 3/20 0.37
RAB9A P51151 1/20 0.37
GAA P10253 1/20 0.37
DRD4 P21917 10/20 0.37
DRD3 P35462 3/20 0.37
DRD2 P14416 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADRA2A P08913 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
ADRA2B P18089 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568230 1.00 MCHR1 (0.40) MCHR1KCNH2DPP4DPP7TSHR
SCHEMBL9568178 0.93 MCHR1 (0.39) MCHR1TSHRALDH1A1GAADRD4
SCHEMBL9568177 0.93 MCHR1 (0.39) MCHR1TSHRALDH1A1GAADRD4
SCHEMBL9568082 0.87 TSHR (0.40) MCHR1KCNH2TSHREPHX1CNR1
Hydrochloric Acid SCHEMBL9568249 0.84 ALDH1A1 (0.42) ALDH1A1RAB9AGAALMNAMEN1
SCHEMBL9568147 0.84 ALDH1A1 (0.41) MCHR1KCNH2TSHREPHX1CNR1
SCHEMBL9568142 0.84 ALDH1A1 (0.41) MCHR1KCNH2TSHREPHX1CNR1
SCHEMBL9568079 0.82 TSHR (0.43) MCHR1KCNH2TSHREPHX1CNR1
SCHEMBL9568102 0.81 TSHR (0.39) MCHR1TSHREPHX1CNR1CNR2
SCHEMBL9568097 0.81 TSHR (0.39) MCHR1TSHREPHX1CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574808-A1 Amidine-biphenyl derivatives, process for their production & medical preparation containing them Dr. Karl Thomae GmbH (DE) 1993-12-22 EP disclosed