SCHEMBL9569191

SCHEMBL9569191

Nc1ncc(C2=Cn3cc(C(=O)O)c(=O)c4cc(F)c(F)c(c43)O2)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 6/20 0.46
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
TOP2A P11388 11/20 0.35
TOP2B Q02880 7/20 0.35
PIM1 P11309 1/20 0.34
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 2/20 0.33
POLB P06746 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
HSP90AA1 P07900 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9569192 0.88 TOP1 (0.37) TOP1CYP3A4CYP2C9
SCHEMBL9509558 0.80 TOP1 (0.52) TOP1TOP2ATOP2BKDM4EALDH1A1
SCHEMBL9509708 0.74 TOP1 (0.52) TOP1TOP2ATOP2BKDM4EKMT2A
SCHEMBL9560362 0.72 TOP1 (0.49) TOP1TOP2ATOP2BKDM4EKMT2A
SCHEMBL9560538 0.71 TOP1 (0.45) TOP1TOP2ATOP2BKDM4EALDH1A1
SCHEMBL9569194 0.71 TOP1 (0.51) TOP1TOP2ATOP2BKDM4EKMT2A
SCHEMBL21729417 0.71 TOP2A (0.69) TOP2ATOP2BKDM4EKMT2AALDH1A1
SCHEMBL14754070 0.69 TOP2A (0.58) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL10538537 0.68 STAT3 (0.47) TOP1PIM1KDM4EKMT2AALDH1A1
SCHEMBL17040509 0.68 TOP2A (0.45) CYP3A4CYP2C9TOP2ATOP2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563734-A1 9-fluoro-7-oxo-7H-pyrido(1,2,3-de)(1,4)benzoxazine carboxylic acids and esters and their use as antiviral agents BAYER AG (DE) 1993-10-06 EP disclosed