SCHEMBL9569720

SCHEMBL9569720

O=C(NC(Cc1ccccc1)C(F)(F)F)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 5/20 0.51
CPA1 P15085 1/20 0.47
ACE P12821 2/20 0.47
NPSR1 Q6W5P4 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CES1 P23141 1/20 0.44
CTSL P07711 1/20 0.44
CYP1A2 P05177 1/20 0.43
FPR2 P25090 1/20 0.42
ECE1 P42892 1/20 0.42
EGFR P00533 1/20 0.41
SRC P12931 1/20 0.41
ALPI P09923 1/20 0.41
PKM P14618 1/20 0.41
PTGS1 P23219 1/20 0.41
XIAP P98170 1/20 0.41
SLC7A5 Q01650 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18765662 0.86 CTRB1 (0.54) CTRB1CPA1ACENPSR1NPC1
SCHEMBL639626 0.83 CTRB1 (0.71) CTRB1CPA1ACENPC1RAB9A
SCHEMBL639902 0.81 ALDH1A1 (0.59) CTRB1CPA1ACENPC1RAB9A
SCHEMBL18793922 0.81 CTRB1 (0.59) CTRB1CPA1ACENPC1RAB9A
SCHEMBL5180357 0.80 NPSR1 (0.69) CPA1ACENPSR1FPR2ECE1
SCHEMBL8613833 0.80 NPSR1 (0.69) CPA1ACENPSR1FPR2ECE1
SCHEMBL8420771 0.80 NPC1 (0.67) CTRB1NPC1RAB9A
SCHEMBL5180354 0.80 NPSR1 (0.69) CPA1ACENPSR1FPR2ECE1
SCHEMBL3533337 0.80 CPA1 (0.47) CTRB1CPA1ACENPSR1NPC1
SCHEMBL4462033 0.80 NPC1 (0.67) CTRB1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5204471-A α-trifluoromethyl-substituted, saturated bicyclic amines BAYER AKTIENGESELLSCHAFT (DE) 1993-04-20 US disclosed
EP-0527385-A1 Alpha-trifluoromethyl substituted, saturated bicyclic amines and process for their preparation BAYER AG (DE) 1993-02-17 EP disclosed