SCHEMBL9574239

SCHEMBL9574239

CCCCCC(Br)OCCCCCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.48
HTR2A P28223 1/20 0.46
PTGES O14684 2/20 0.43
ALOX5 P09917 2/20 0.43
PPARG P37231 2/20 0.43
SIGMAR1 Q99720 5/20 0.42
CSNK1E P49674 1/20 0.41
PLA2G10 O15496 1/20 0.41
PLA2G1B P04054 1/20 0.41
PLA2G2A P14555 1/20 0.41
PLA2G5 P39877 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028474 0.81 CETP (0.45) CSNK1E
SCHEMBL22922951 0.81 KCNH2 (0.47) KCNH2HTR2APTGESALOX5PPARG
SCHEMBL25065427 0.81 KCNH2 (0.47) KCNH2HTR2APTGESALOX5PPARG
SCHEMBL4749538 0.81 KCNH2 (0.51) KCNH2HTR2ASIGMAR1CSNK1E
SCHEMBL2854089 0.81 KCNH2 (0.51) KCNH2HTR2ASIGMAR1CSNK1E
SCHEMBL7062802 0.79 SIGMAR1 (0.49) KCNH2HTR2ASIGMAR1CSNK1E
SCHEMBL7797335 0.78 CSNK1E (0.44) KCNH2HTR2APTGESALOX5PPARG
SCHEMBL11785905 0.78 SIGMAR1 (0.50) KCNH2HTR2ASIGMAR1L3MBTL1
SCHEMBL19322733 0.77 KCNH2 (0.59) KCNH2HTR2ASIGMAR1TDP1L3MBTL1
SCHEMBL22268758 0.77 KCNH2 (0.59) KCNH2HTR2ASIGMAR1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5243076-A Adrenergic stimulant intermediates GLAXO GROUP LTD. 1993-09-07 US disclosed
US-5225445-A Respiratory system disorders GLAXO GROUP LTD. 1993-07-06 US disclosed
US-5091422-A Treating inflammatory or allergic skin disease, lowering gastric acidity GLAXO GROUP LIMITED (GB) 1992-02-25 US disclosed
US-4992474-A Adrenergic stimulants GLAXO GROUP LTD. (GB) 1991-02-12 US disclosed