SCHEMBL9577985

SCHEMBL9577985

O=c1oc(=O)n(C2CC2)c2cc(F)c(F)cc12

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.36
CYP11B1 P15538 4/20 0.35
CYP3A4 P08684 2/20 0.35
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM5 P08912 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
CYP19A1 P11511 1/20 0.33
ADRA2B P18089 1/20 0.33
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31433786 0.88 IRAK4 (0.33) CYP11B2CYP11B1CYP3A4CHRM2CHRM4
SCHEMBL2117902 0.75 MAT2A (0.42) CYP11B2CHRM1
SCHEMBL11853247 0.73 TNKS (0.42) CHRM4CHRM5CHRM1
SCHEMBL4503078 0.71 MPO (0.40) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL4504709 0.71 PGR (0.47) CYP11B2CHRM2CHRM4CHRM5CHRM1
SCHEMBL10846917 0.67 NPSR1 (0.51) CHRM2CHRM4CHRM1CHRM3
SCHEMBL3314661 0.66 PGR (0.54) CHRM2CHRM4CHRM1CHRM3
SCHEMBL3344439 0.66 PGR (0.39)
SCHEMBL9014024 0.65 PRKD3 (0.40) CYP11B2CHRM2CHRM1TOP2ATOP2B
SCHEMBL606349 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0370686-B1 A process for preparing quinolone carboxylic acid intermediates PFIZER (US) 1993-12-29 EP disclosed
US-5064958-A CHEMICAL INTERMEDIATES FOR ANTIBACTERIAL COMPOUNDS PFIZER INC. (US) 1991-11-12 US disclosed
US-4939290-A Bactericides PFIZER INC. (US) 1990-07-03 US disclosed
EP-0370686-A2 A process for preparing quinolone carboxylic acid intermediates PFIZER INC. (US) 1990-05-30 EP disclosed