SCHEMBL957799

SCHEMBL957799

O=P(O)(O)C(CS)P(=O)(O)O

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FDPS P14324 8/20 0.46
ENPEP Q07075 2/20 0.44
KDM4E B2RXH2 1/20 0.39
MMP2 P08253 1/20 0.39
THRB P10828 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TYMS P04818 1/20 0.35
ANPEP P15144 1/20 0.35
ERAP2 Q6P179 1/20 0.35
LMNA P02545 1/20 0.33
LAP3 P28838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8160239 0.83 FDPS (0.44) FDPSENPEP
SCHEMBL250204 0.72 FDPS (0.50) FDPSKDM4EMMP2THRBMAPK1
SCHEMBL10785210 0.72 FDPS (0.67) FDPSKDM4EMMP2THRBMAPK1
SCHEMBL5011508 0.71 FDPS (0.58) FDPSENPEPTYMS
SCHEMBL4124789 0.70
SCHEMBL2455930 0.69 FDPS (0.60) FDPSENPEP
SCHEMBL29449121 0.69 FDPS (0.48) FDPSKDM4EMMP2THRBMAPK1
SCHEMBL3904202 0.69 FDPS (0.48) FDPSKDM4EMMP2THRBMAPK1
SCHEMBL8713308 0.69 FDPS (0.48) FDPSKDM4EMMP2THRBMAPK1
SCHEMBL56898 0.69 FDPS (0.48) FDPSKDM4EMMP2THRBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689861-B2 POLYURETHANE HAVING A GEMINAL BISPHOSPHONATE SUBSTITUENT PENDANT THE CHILDREN'S HOSPITAL OF PHILADELPHI 2004-02-10 US claimed
US-20230348785-A1 FLAME RETARDANT FOR WOODY MATERIALS AND FLAME-RETARDANT WOODY MATERIAL DAIHACHI CHEM IND (JP) 2023-11-02 US disclosed
US-11760936-B2 Flame retardant for woody materials and flame-retardant woody material DAIHACHI CHEMICAL INDUSTRY CO., LTD. (JP) 2023-09-19 US disclosed
CN-115011360-A Flame retardant for wood material and flame-retardant wood material 大八化学工业株式会社 2022-09-06 CN disclosed
CN-110678533-B Flame retardant for wood material and flame-retardant wood material 大八化学工业株式会社 2022-07-08 CN disclosed
US-20210147750-A1 FLAME RETARDANT FOR WOODY MATERIALS AND FLAME-RETARDANT WOODY MATERIAL DAIHACHI CHEMICAL INDUSTRY CO., LTD. (JP) 2021-05-20 US disclosed
EP-3633012-A1 FLAME RETARDANT FOR WOODY MATERIALS AND FLAME-RETARDANT WOODY MATERIAL Daihachi Chemical Industry Co., Ltd. (JP) 2020-04-08 EP disclosed
CN-110678533-A Flame retardant for wood material and flame-retardant wood material 大八化学工业株式会社 2020-01-10 CN disclosed
US-20120184941-A1 MULTICOMPONENT MAGNETIC NANOPARTICLE DELIVERY SYSTEM FOR LOCAL DELIVERY TO HEART VALVE LEAFLETS AND OTHER ANIMAL TISSUES The Children's Hosital of Philadelphia (US) 2012-07-19 US disclosed
EP-2456500-A1 A MULTICOMPONENT MAGNETIC NANOPARTICLE DELIVERY SYSTEM FOR LOCAL DELIVERY TO HEART VALVE LEAFLETS AND OTHER ANIMAL TISSUES The Children's Hospital of Philadelphia (US) 2012-05-30 EP disclosed
EP-1208129-A2 2002-05-29 EP disclosed
US-6320011-B1 POLYURETHANE HAVING A GEMINAL BISPHOSPHONATE SUBSTITUENT PENDANT THEREFROM; IMPLANTABLE DEVICES THAT ARE CALCIFICATION-RESISTANT, THROMBOGENESIS-RESISTANT, AND DEGRADATION-RESISTANT THE CHILDREN'S HOSPITAL OF PHILADELPHIA 2001-11-20 US disclosed
WO-2001008123-A1 DERIVATIZED POLYURETHANE COMPOSITIONS AND METHODS OF MAKING THE CHILDREN'S HOSPITAL OF PHILADELPHIA (US) 2001-02-01 WO disclosed
EP-0650361-B1 COMPOSITIONS FOR THE TREATMENT OF ARTHRITIS CONTAINING PHOSPHONATES AND NSAIDS PROCTER & GAMBLE PHARMA (US) 1999-04-28 EP disclosed
US-5869471-A Methods for the treatment of arthritis using phosphonates and NSAIDS THE PROCTOR & GAMBLE COMPANY (US) 1999-02-09 US disclosed
EP-0650361-A1 COMPOSITIONS FOR THE TREATMENT OF ARTHRITIS CONTAINING PHOSPHONATES AND NSAIDS PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1995-05-03 EP disclosed
WO-1994000130-A1 COMPOSITIONS FOR THE TREATMENT OF ARTHRITIS CONTAINING PHOSPHONATES AND NSAIDS PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1994-01-06 WO disclosed
US-4810486-A FROM SULFONATE-CONTAINING BIS-PHOSPHONIC ACID, REDUCING AGENT, PERTECHNEATATE IONS AMERSHAM INTERNATIONAL PLC. (GB) 1989-03-07 US disclosed
EP-0270648-A1 BONE-SEEKING COMPLEXES OF TECHNETIUM-99m AMERSHAM INTERNATIONAL plc (GB) 1988-06-15 EP disclosed
WO-1988000061-A1 BONE-SEEKING COMPLEXES OF TECHNETIUM-99m AMERSHAM INTERNATIONAL PLC (GB) 1988-01-14 WO disclosed