SCHEMBL9583296

SCHEMBL9583296

CSc1ncnc2c1ncn2C(O)OCCCO

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.46
TSHR P16473 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.43
TP53 P04637 1/20 0.43
ADA P00813 4/20 0.35
PDE2A O00408 3/20 0.35
CYP3A4 P08684 2/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HIF1A Q16665 1/20 0.35
LMNA P02545 1/20 0.34
BLM P54132 1/20 0.34
ADORA2A P29274 3/20 0.34
ADORA2B P29275 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9583319 0.82 HK1 (0.41) CYP1A2
SCHEMBL9583681 0.81 ADORA2A (0.55) CYP1A2TSHRSMN1; SMN2ADAPDE2A
SCHEMBL10540197 0.80 CDK2 (0.36) CYP1A2TSHRPDE4D
SCHEMBL9584677 0.80 CYP1A2 (0.48) CYP1A2
SCHEMBL9583194 0.80 YTHDC1 (0.47) ADORA1AHCY
SCHEMBL6363954 0.73 ADORA2A (0.60) CYP1A2TSHRSMN1; SMN2TP53ADORA2A
SCHEMBL9583624 0.73 CYP1A2 (0.40) CYP1A2TSHRSMN1; SMN2TP53
SCHEMBL8466930 0.71 CYP1A2 (0.72) CYP1A2TSHRSMN1; SMN2TP53ALDH1A1
SCHEMBL8839827 0.71 FDPS (0.40) CYP1A2CYP3A4ALDH1A1HSD17B10
SCHEMBL18521260 0.71 CYP1A2 (0.49) CYP1A2TSHRSMN1; SMN2TP53ADA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5250535-A Herpes virus; nontoxic; side effect reduction; humans and veterinary medicine SYNTEX INC. (US) 1993-10-05 US disclosed
US-4803271-A Process for preparing guanine derivatives SYNTEX (U.S.A.) INC. (US) 1989-02-07 US disclosed
EP-0105135-B1 SUBSTITUTED 9-(1-0- OR 3-0-MONOSUBSTITUTED OR 1,3-DI-0-SUBSTITUTED 1,3 DIHYDROXY-2-PROPOXYMETHYL) PURINES AS ANTIVIRAL AGENTS SYNTEX (U.S.A.) INC. (US) 1987-03-18 EP disclosed
US-4612314-A Substituted 9-(1 or 3-monoacyloxy or 1,3-diacyloxy-2-propoxymethyl) purines as antiviral agent SYNTEX (U.S.A.) INC. (US) 1986-09-16 US disclosed
US-4609661-A HERPES VIRUS SYNTEX (U.S.A.) INC. (US) 1986-09-02 US disclosed
US-4556659-A Substituted 9-(1-0- or 3-0-monosubstituted or 1,3-Di-0-substituted propoxymethyl)-purines as antiviral agents SYNTEX (U.S.A.) INC. (US) 1985-12-03 US disclosed
EP-0105135-A1 Substituted 9-(1-0- or 3-0-monosubstituted or 1,3-di-0-substituted 1,3 dihydroxy-2-propoxymethyl) purines as antiviral agents SYNTEX (U.S.A.) INC. (US) 1984-04-11 EP disclosed
EP-0085424-A2 Substituted 9-(1 or 3-monoacyloxy or 1,3-diacyloxy-2-propoxymethyl)purines as antiviral agent SYNTEX (U.S.A.) INC. (US) 1983-08-10 EP disclosed