SCHEMBL9587488

SCHEMBL9587488

CNc1nc(N)c2cc(N(C)Cc3ccc(S(=O)(=O)c4ccccc4)cc3)ccc2n1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.45
TYMS P04818 3/20 0.44
IP6K1 Q92551 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9586795 0.89 TRIM58 (0.46) TYMSIP6K1
SCHEMBL1065778 0.87 DHFR (0.59) DHFRTYMS
SCHEMBL9587910 0.86 DHFR (0.47) DHFRTYMSIP6K1
SCHEMBL9587723 0.84 DHFR (0.45) DHFRTYMSIP6K1
SCHEMBL9587516 0.82 IP6K1 (0.40) TYMSIP6K1
SCHEMBL9586237 0.81 DHFR (0.59) DHFR
SCHEMBL9587848 0.81 DHFR (0.57) DHFR
SCHEMBL9587020 0.80 DHFR (0.45) DHFRTYMSIP6K1
SCHEMBL9587570 0.79 DHFR (0.57) DHFR
SCHEMBL9587214 0.79 DHFR (0.57) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013079-A1 ANTIFOLATE QUINAZOLINES AGOURON PHARMACEUTICALS, INC. (US) 1993-07-08 WO disclosed