SCHEMBL9587516

SCHEMBL9587516

CNc1ncc2cc(N(C)Cc3ccc(S(=O)(=O)c4ccccc4)cc3)ccc2n1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.40
NAMPT P43490 6/20 0.40
TYMS P04818 4/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
PIK3CA P42336 2/20 0.36
RPS6KB1 P23443 1/20 0.36
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9586795 0.83 TRIM58 (0.46) IP6K1NAMPTTYMSPTGDR2
SCHEMBL9587488 0.82 DHFR (0.45) IP6K1TYMS
SCHEMBL9587514 0.77 CA1 (0.44) NAMPT
SCHEMBL1065778 0.73 DHFR (0.59) TYMS
SCHEMBL9587910 0.72 DHFR (0.47) IP6K1TYMS
SCHEMBL9587020 0.72 DHFR (0.45) IP6K1TYMS
SCHEMBL9586297 0.71 DHFR (0.45) IP6K1TYMS
SCHEMBL9587730 0.71 DHFR (0.55) IP6K1TYMS
SCHEMBL9587180 0.70 IP6K1 (0.44) IP6K1TYMS
SCHEMBL9587723 0.70 DHFR (0.45) IP6K1TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013079-A1 ANTIFOLATE QUINAZOLINES AGOURON PHARMACEUTICALS, INC. (US) 1993-07-08 WO disclosed