SCHEMBL9588205

SCHEMBL9588205

c1ccc2c3c(cnc2c1)OCCN3

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.40
KDM4E B2RXH2 2/20 0.38
GPR3 P46089 1/20 0.38
ADRA2A P08913 2/20 0.36
ADRA2C P18825 2/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
NCF1 P14598 2/20 0.36
ADRB2 P07550 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
GRM1 Q13255 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
HSD17B10 Q99714 2/20 0.34
RHOA P61586 1/20 0.34
GLA P06280 1/20 0.34
HPGD P15428 1/20 0.34
ADRA2B P18089 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23405733 0.91 KDM4E (0.36) GRM5KDM4EGPR3NCF1ADRB2
SCHEMBL30079947 0.91 KDM4E (0.36) GRM5KDM4EGPR3NCF1ADRB2
SCHEMBL25666745 0.79 LMNA (0.37) GRM5KDM4EADRA2AADRA2CADRA1D
SCHEMBL9590061 0.79 GRM1 (0.41) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL13652212 0.76 NCF1 (0.44) KDM4EADRA1DADRA1AADRA1BNCF1
SCHEMBL30079880 0.75 KDM4E (0.36) KDM4EGPR3NCF1ADRB2ALDH1A1
SCHEMBL25666758 0.75 KDM4E (0.36) KDM4EGPR3NCF1ADRB2ALDH1A1
SCHEMBL22744581 0.75 SSTR4 (0.36) GRM5KDM4EGPR3NCF1ADRB2
SCHEMBL1191697 0.74 KDM4E (0.38) GRM5KDM4EGPR3NCF1ADRB2
SCHEMBL25666734 0.73 KDM4E (0.42) KDM4EGPR3ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4743601-A MEMORY ENHANCEMENT HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-05-10 US claimed
WO-2023109909-A1 AROMATIC HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND USES THEREOF 上海翊石医药科技有限公司 2023-06-22 WO disclosed
US-11512095-B2 BCL6 inhibitors THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2022-11-29 US disclosed
US-5182275-A Intermediates for memory enhancers HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-26 US disclosed
US-4942168-A INTERMEDIATES FOR 1,2-DIHYDRO-3-METHYL-3H-1,4-OXAZINO 2,3-C!QU INOLINE HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-07-17 US disclosed
EP-0299345-A3 Dihydro-1,4-oxazino(2,3-c)quinolines, a process and intermediates for the preparation thereof and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1990-06-13 EP disclosed
EP-0299345-A2 Dihydro-1,4-oxazino(2,3-c)quinolines, a process and intermediates for the preparation thereof and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-01-18 EP disclosed
EP-0299345-A2 Dihydro-1,4-oxazino(2,3-c)quinolines, a process and intermediates for the preparation thereof and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-01-18 EP disclosed
US-4743601-A MEMORY ENHANCEMENT HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-05-10 US disclosed
US-4743601-A MEMORY ENHANCEMENT HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11512095-B2 BCL6 inhibitors BCL6, BCL6B, BCL3 GRM5 4476/4885KDM4E 481/4885GPR3 3754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.