SCHEMBL9591998

SCHEMBL9591998

CCCCc1nc(Br)c(P(=O)(O)O)n1COCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
CETP P11597 3/20 0.40
ALDH1A1 P00352 1/20 0.39
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
AGTR1 P30556 2/20 0.38
AGTR2 P50052 2/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
GLA P06280 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9593156 0.83 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL9584286 0.79
SCHEMBL29954342 0.72 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DTLR8
SCHEMBL9592123 0.71
SCHEMBL6928223 0.70 ALDH1A1 (0.45) ALDH1A1TLR7LMNAMAPK1
SCHEMBL6922966 0.68 ALDH1A1 (0.43) ALDH1A1TLR7LMNAMAPK1
SCHEMBL8532701 0.67 ALDH1A1 (0.42) ALDH1A1LMNAMAPK1
SCHEMBL8536161 0.66 ALDH1A1 (0.43) ALDH1A1LMNAMAPK1
SCHEMBL8536407 0.64 ALDH1A1 (0.46) ALDH1A1LMNAMAPK1
Butylbenzyl SCHEMBL4983622 0.63 CETP (0.64) CETPALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208235-A Phosphonic or phosphinic acid derivatives as inhibitors of angiotnesin II for cardiovascular disorders and hypotensives E. R. SQUIBB & SONS, INC. (US) 1993-05-04 US disclosed