SCHEMBL9596607

SCHEMBL9596607

O=C(O)C=CC(=O)ON1CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.39
KDM4E B2RXH2 1/20 0.37
CYP3A4 P08684 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TSHR P16473 2/20 0.35
TP53 P04637 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
EGLN3 Q9H6Z9 1/20 0.35
CA2 P00918 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
PMP22 Q01453 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CHKA P35790 1/20 0.31
HRH1 P35367 1/20 0.31
ATM Q13315 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9596598 1.00 HCAR2 (0.39) HCAR2KDM4ECYP3A4HSD17B10TSHR
Water SCHEMBL28189169 0.98 HCAR2 (0.38) HCAR2KDM4ECYP3A4HSD17B10TSHR
SCHEMBL28719611 0.98 HCAR2 (0.38) HCAR2KDM4ECYP3A4HSD17B10TSHR
SCHEMBL5874482 0.92 CA2 (0.37) CA2CA12CA1CA9CHKA
SCHEMBL5874850 0.92 CA2 (0.37) CA2CA12CA1CA9CHKA
Pyridine SCHEMBL28100292 0.87 KDM4E (0.39) HCAR2KDM4ECYP3A4HSD17B10ALDH1A1
SCHEMBL3632775 0.82 HCAR2 (0.43) HCAR2KDM4ETSHRTP53EGLN1
SCHEMBL10992799 0.82 HCAR2 (0.43) HCAR2KDM4ETSHRTP53EGLN1
SCHEMBL10859682 0.80 HCAR2 (0.41) HCAR2TSHRTP53EGLN1EGLN3
SCHEMBL29040960 0.80 CA12 (0.30) CA2CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5183902-A Muscle relaxants A. H. ROBINS COMPANY, INCORPORATED (US) 1993-02-02 US disclosed
US-5068231-A Ureas and thioureas for relaxing muscles A. H. ROBINS COMPANY INCORPORATED (US) 1991-11-26 US disclosed
US-4956359-A CARBOXAMIDES OR THIOCARBOXAMIDES OF ARYL OXY OR THIO AZETIDINES A. H. ROBINS COMPANY, INC. (US) 1990-09-11 US disclosed