SCHEMBL9599601

SCHEMBL9599601

CCCCCN1CCc2ccccc2C1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.51
OPRK1 P41145 1/20 0.51
ACE P12821 4/20 0.50
HDAC8 Q9BY41 3/20 0.50
HDAC3 O15379 2/20 0.50
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
NCOR2 Q9Y618 2/20 0.50
PRCP P42785 1/20 0.47
KCNH2 Q12809 1/20 0.42
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4239790 0.85 PRCP (0.60) ACEHDAC8HDAC3HDAC1HDAC2
SCHEMBL3609218 0.79 ACE (0.70) ACEHDAC3HDAC1
SCHEMBL3609137 0.78 ACE (0.52) ACEHDAC8HDAC3HDAC1HDAC2
SCHEMBL22525235 0.77 PRCP (0.57) OPRM1OPRK1ACEPRCP
SCHEMBL2088793 0.77 PRCP (0.57) OPRM1OPRK1ACEPRCP
SCHEMBL9387516 0.77 OPRM1 (0.57) OPRM1OPRK1HDAC8HDAC3HDAC1
SCHEMBL28851671 0.77 CYP2D6 (0.47) OPRM1OPRK1HDAC8HDAC3HDAC1
SCHEMBL29159488 0.77 OPRM1 (0.54) OPRM1OPRK1HDAC8HDAC3HDAC1
SCHEMBL3612877 0.76 OPRM1 (0.42) OPRM1OPRK1HDAC8HDAC3HDAC1
SCHEMBL3608890 0.76 OPRM1 (0.44) OPRM1OPRK1HDAC8HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5238935-A Treating atherosclerosis SCHERING CORPORATION (US) 1993-08-24 US disclosed
EP-0514851-A1 N-acyl-tetrahydroisoquinolines as inhibitors of acyl-coenzyme a:cholesterol acyl transferase SCHERING CORPORATION (US) 1992-11-25 EP disclosed
US-5124337-A Treating atherosclerosis SCHERING CORPORATION (US) 1992-06-23 US disclosed