SCHEMBL9387516

SCHEMBL9387516

CCCCN1CCc2ccccc2C1NC(=O)O

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.57
OPRK1 P41145 3/20 0.57
HDAC8 Q9BY41 5/20 0.48
HDAC1 Q13547 4/20 0.48
HDAC2 Q92769 4/20 0.48
HDAC3 O15379 3/20 0.48
NCOR2 Q9Y618 3/20 0.48
PRCP P42785 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
SIGMAR1 Q99720 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9387259 0.92 OPRM1 (0.48) OPRM1OPRK1HDAC8HDAC1HDAC2
SCHEMBL11055845 0.89 OPRM1 (0.53) OPRM1OPRK1HDAC8HDAC1HDAC2
SCHEMBL11051207 0.81 HTR1A (0.46) OPRM1OPRK1HDAC8HDAC1HDAC2
SCHEMBL9599601 0.77 OPRM1 (0.51) OPRM1OPRK1HDAC8HDAC1HDAC2
SCHEMBL20788100 0.73 OPRM1 (1.00) OPRM1OPRK1L3MBTL1
SCHEMBL28851671 0.72 CYP2D6 (0.47) OPRM1OPRK1HDAC8HDAC1HDAC2
Hexane SCHEMBL28019996 0.72 EPHX2 (0.56) L3MBTL1
SCHEMBL8560553 0.70 OPRM1 (0.49) OPRM1OPRK1HDAC8HDAC1HDAC2
SCHEMBL2358733 0.70 MTNR1A (0.40) OPRM1OPRK1HDAC8HDAC1HDAC2
SCHEMBL29159488 0.69 OPRM1 (0.54) OPRM1OPRK1HDAC8HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538248-A4 1994-08-03 EP claimed
EP-0538248-A1 TETRAHYDROISOQUINOLINYLCARBAMATES OF 1,2,3,3A,8,8A-HEXAHYDRO-1,3A,8-TRIMETHYLPYRROLO [2,3-B]INDOLE HOECHST MARION ROUSSEL, INC. (US) 1993-04-28 EP claimed