SCHEMBL9601697

SCHEMBL9601697

Cn1nccc1NCCC[O]

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 2/20 0.40
AVPR1A P37288 2/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.37
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.34
COMT P21964 1/20 0.33
CTSK P43235 1/20 0.33
HPGDS O60760 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
CYP1A2 P05177 1/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
LRRK2 Q5S007 1/20 0.31
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27625405 0.84 CYP1A2 (0.44) OXTRAVPR1ARAB9AKMT2AL3MBTL1
SCHEMBL4036017 0.78 OXTR (0.38) OXTRAVPR1ARAB9AKMT2APOLB
SCHEMBL22957177 0.78 OXTR (0.38) OXTRAVPR1ARAB9AKMT2APOLB
SCHEMBL26091092 0.76 POLB (0.47) OXTRAVPR1ARAB9AKMT2APOLB
SCHEMBL4032778 0.73
SCHEMBL12763786 0.70 POLB (0.38) OXTRAVPR1ARAB9AKMT2APOLB
SCHEMBL14937937 0.68 KCNN1 (0.50) RAB9AKMT2APOLB
SCHEMBL309844 0.68
SCHEMBL21383369 0.67 KMT2A (0.55) OXTRAVPR1ARAB9AKMT2APOLB
Hydrochloric Acid SCHEMBL21248629 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0232623-B1 1-CARBACEPHALOSPORIN ANTIBIOTICS ELI LILLY AND COMPANY (US) 1993-03-17 EP disclosed
US-4892942-A 1-CARBA (DETHIA)CEPHALOSPORINS ELI LILLY AND COMPANY (US) 1990-01-09 US disclosed
US-4791106-A 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1988-12-13 US disclosed
EP-0232623-A1 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1987-08-19 EP disclosed