SCHEMBL9602154

SCHEMBL9602154

CN1CCN(C=O)C(=O)C1=O

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
BRD4 O60885 1/20 0.31
BRD2 P25440 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27666999 0.81 BRD4 (0.31) BRD4BRD2
SCHEMBL717518 0.79 BRD4 (0.43) MEN1KMT2ABRD4BRD2
SCHEMBL11138071 0.78
SCHEMBL9600407 0.73 GRM5 (0.35)
SCHEMBL9602860 0.71 SMN1; SMN2 (0.37)
SCHEMBL9600719 0.70 PLA2G2A (0.38) MEN1KMT2A
SCHEMBL9600841 0.68 PLA2G2A (0.44)
SCHEMBL27877993 0.68 SMN1; SMN2 (0.31)
SCHEMBL14428797 0.68 BRD4 (0.52) MEN1KMT2ABRD4BRD2
SCHEMBL2561381 0.67 PIK3CD (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4283333-A α-[4-Oxoazetidin-1-yl]-acetic acid compounds useful as intermediates in preparing 1-oxadethiacephalosporins SHIONOGI & CO., LTD. (JP) 1981-08-11 US claimed
US-4066641-A METHOD FOR CYCLIZATION TO GIVE CEPHEM RING HAMASHIMA YOSHIO 1978-01-03 US claimed
EP-0215435-B1 2-OXA-ISOCEPHEM COMPOUNDS, COMPOSITIONS CONTAINING SAME AND PROCESSES FOR PREPARING SAME OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-03-03 EP disclosed
US-4831026-A ANTIBIOTICS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-05-16 US disclosed
EP-0215435-A1 2-Oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-03-25 EP disclosed
US-4283333-A α-[4-Oxoazetidin-1-yl]-acetic acid compounds useful as intermediates in preparing 1-oxadethiacephalosporins SHIONOGI & CO., LTD. (JP) 1981-08-11 US disclosed
US-4269773-A CEPHALOSPORINS SHIONOGI & CO., LTD. (JP) 1981-05-26 US disclosed
US-4223132-A Selective conversion of benzyl alcohol carboxylates to the free acid form SHIONOGI & CO., LTD. (JP) 1980-09-16 US disclosed
US-4159984-A METAL AND PROTON DONOR SHIONOGI & CO., LTD. (JP) 1979-07-03 US disclosed
US-4066641-A METHOD FOR CYCLIZATION TO GIVE CEPHEM RING HAMASHIMA YOSHIO 1978-01-03 US disclosed