SCHEMBL9602346

SCHEMBL9602346

O=C(Cc1cccnc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 5/20 0.61
TSHR P16473 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
TBXAS1 P24557 2/20 0.53
TBXA2R P21731 1/20 0.53
NAMPT P43490 2/20 0.52
CES2 O00748 1/20 0.50
ALOX15 P16050 1/20 0.50
CASP1 P29466 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50
NAPRT Q6XQN6 1/20 0.49
ALDH1A1 P00352 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
SORT1 Q99523 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602354 0.89 MEN1 (0.57) VNN1TSHRMEN1KMT2ATBXAS1
SCHEMBL11792850 0.85 VNN1 (0.58) VNN1MEN1KMT2ANAMPTNAPRT
SCHEMBL2929610 0.85 VNN1 (0.57) VNN1TSHRMEN1KMT2ANAMPT
SCHEMBL6970291 0.84 CES2 (0.61) MEN1KMT2ACES2ALDH1A1DDR1
SCHEMBL28977515 0.83 VNN1 (0.54) VNN1TSHRMEN1KMT2ANAMPT
SCHEMBL423798 0.83 DDR1 (0.59) VNN1MEN1KMT2ACES2RAB9A
SCHEMBL11626058 0.81 VNN1 (0.67) VNN1TSHRMEN1KMT2ANAMPT
Hydrochloric Acid SCHEMBL11627866 0.80 VNN1 (0.65) VNN1TSHRMEN1KMT2ANAMPT
SCHEMBL17672056 0.79 NAPRT (0.65) MEN1KMT2ANAPRTALDH1A1RAB9A
SCHEMBL31326722 0.79 NAPRT (0.65) MEN1KMT2ANAPRTALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221601-B1 [[[(3-Pyridinyl)methylen]amino]oxy]alkanoic acids and esters JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-10 EP disclosed
US-5180832-A Chemical intermediate for thromboxane A2 inhibitor JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-19 US disclosed
US-4746671-A THROMBOXANE SYNTHETASE INHIBITION JANSSEN PHARMACEUTICA N.V. (BE) 1988-05-24 US disclosed