SCHEMBL9602508

SCHEMBL9602508

CCOC(=O)c1cc(CCO)ccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.47
CYP4A11 Q02928 3/20 0.47
CYP1A2 P05177 1/20 0.46
GABRA1 P14867 7/20 0.44
GABRG2 P18507 7/20 0.44
GABRB3 P28472 7/20 0.44
GABRA5 P31644 7/20 0.44
GABRA3 P34903 7/20 0.44
GABRA2 P47869 7/20 0.44
GABRA4 P48169 7/20 0.44
GABRA6 Q16445 7/20 0.44
GABRP O00591 6/20 0.44
GABRD O14764 6/20 0.44
GABRB1 P18505 6/20 0.44
GABRB2 P47870 6/20 0.44
GABRE P78334 6/20 0.44
GABRG1 Q8N1C3 6/20 0.44
GABRG3 Q99928 6/20 0.44
GABRQ Q9UN88 6/20 0.44
CDC7 O00311 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2935704 0.88 CYP1A2 (0.49) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL9518746 0.84 CYP4A11 (0.54) CYP4F2CYP4A11ALDH1A1KDM4EMAPK1
SCHEMBL7008579 0.83 CYP1A2 (0.47) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL128612 0.83 CYP1A2 (0.47) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL480291 0.83 CYP4F2 (0.52) CYP4F2CYP4A11CYP1A2GABRA1GABRG2
Hydrochloric Acid SCHEMBL20357239 0.82 CYP1A2 (0.46) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL744204 0.80 GABRA1 (0.43) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL743703 0.79 CYP1A2 (0.44) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL127699 0.79 CYP1A2 (0.53) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL13813279 0.79 ALDH1A1 (0.44) CYP4F2CYP4A11GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5217963-A Antiischemic, antiepileptic agent CIBA-GEIGY CORPORATION (US) 1993-06-08 US disclosed
US-5057506-A Anticonvulsants, antispasmodic and antischemic agents CIBA-GEIGY CORPORATION (US) 1991-10-15 US disclosed
US-4906621-A Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade CIBA-GEIGY CORPORATION (US) 1990-03-06 US disclosed
US-4898854-A NERVOUS SYSTEM DISORDERS CIBA-GEIGY CORPORATION (US) 1990-02-06 US disclosed