SCHEMBL9602840

SCHEMBL9602840

C=CC(Br)c1csc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.42
ALOX5 P09917 1/20 0.41
MAPT P10636 3/20 0.38
CMA1 P23946 1/20 0.37
SLC6A2 P23975 3/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KCNH2 Q12809 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5826470 0.82 CYP2A6 (0.50) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL28679598 0.79 ALOX5 (0.46) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL30061208 0.79 CYP2A6 (0.46) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL15596088 0.79 CYP2A6 (0.46) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL19682789 0.76 ALOX5 (0.51) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL9281496 0.72 ALOX5 (0.44) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL9634797 0.71 ALDH1A1 (0.36) CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL717441 0.71 ALOX5 (0.54) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL6026188 0.71 ALOX5 (0.46) CYP2A6ALOX5MAPTCMA1SLC6A2
SCHEMBL13920405 0.68 ALOX5 (0.42) CYP2A6ALOX5MAPTCMA1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279263-B1 INDOLE, BENZOFURAN, BENZOTHIOPHENE CONTAINING LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1993-08-04 EP disclosed
US-4873259-A Indole, benzofuran, benzothiophene containing lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1989-10-10 US disclosed
EP-0279263-A2 Indole, benzofuran, benzothiophene containing lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1988-08-24 EP disclosed