SCHEMBL9604500

SCHEMBL9604500

Cc1cc(C)c2c(c1)N=C(C(=O)O)NS2(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 3/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA4 P22748 2/20 0.42
CA7 P43166 2/20 0.42
KDM4E B2RXH2 1/20 0.33
TPMT P51580 1/20 0.32
HCAR2 Q8TDS4 1/20 0.31
GPR17 Q13304 1/20 0.31
ALPL P05186 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9604869 0.73 CA2 (0.42) CA9CA12CA1CA2CA4
SCHEMBL20777728 0.64 CA2 (0.36) CA9CA12CA1CA2CA4
SCHEMBL11677692 0.61 CA12 (0.54) CA9CA12CA1CA2CA4
SCHEMBL7773292 0.59 TTR (0.42) CA9CA12CA1CA2CA4
SCHEMBL21870 0.57 KDM4E (0.55) KDM4ETPMT
SCHEMBL377596 0.57 KDM4E (0.55) KDM4ETPMT
SCHEMBL17558193 0.56 KDM4E (0.53) KDM4ETPMT
SCHEMBL6912557 0.56 KDM4E (0.53) KDM4ETPMT
SCHEMBL6917032 0.56 KDM4E (0.53) KDM4ETPMT
SCHEMBL6915449 0.56 KDM4E (0.53) KDM4ETPMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993021171-A1 USE OF 2H-1,2,4-BENZOTHIADIAZINE-1,1-DIOXIDE-3-CARBOXYLIC ACID DERIVATIVES FOR PREPARING NMDA/AMPA RECEPTOR ANTAGONIST DRUGS, NOVEL PRODUCTS, PREPARATION THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1993-10-28 WO disclosed