SCHEMBL9604540

SCHEMBL9604540

O=C1CN2C(=O)C(=O)c3ccccc3C2=N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.47
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
GAA P10253 2/20 0.43
CASP3 P42574 2/20 0.40
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
CDC25B P30305 1/20 0.38
MAPT P10636 3/20 0.37
HPGD P15428 2/20 0.37
CES1 P23141 4/20 0.37
MAOA P21397 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
PPARG P37231 2/20 0.37
CES2 O00748 1/20 0.37
APAF1 O14727 1/20 0.37
TERT O14746 1/20 0.37
PLIN1 O60240 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10465075 0.89 CYP2D6 (0.56) CYP2D6ALDH1A1KDM4ESMN1; SMN2GAA
SCHEMBL9873658 0.71 CYP2D6 (0.54) CYP2D6ALDH1A1KDM4ESMN1; SMN2GAA
SCHEMBL9868719 0.71 ALDH1A1 (0.43) ALDH1A1KDM4ESMN1; SMN2GAAKMT2A
SCHEMBL9414994 0.62 KDM4E (0.41) CYP2D6ALDH1A1KDM4ESMN1; SMN2GAA
SCHEMBL11604852 0.60 SIGMAR1 (0.58) KDM4ESMN1; SMN2GAAKMT2AMEN1
Anthraquinone SCHEMBL1901249 0.60 MEN1 (1.00) CYP2D6ALDH1A1KDM4ESMN1; SMN2CASP3
Anthraquinone SCHEMBL14943 0.60 MEN1 (1.00) CYP2D6ALDH1A1KDM4ESMN1; SMN2CASP3
Anthraquinone SCHEMBL29358690 0.60 MEN1 (1.00) CYP2D6ALDH1A1KDM4ESMN1; SMN2CASP3
SCHEMBL2493946 0.59 DNMT1 (0.62) KMT2AMEN1DNMT1
SCHEMBL9159989 0.59 NPC1 (0.45) ALDH1A1KDM4ESMN1; SMN2GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0205879-B1 PROCESS FOR THE PREPARATION OF HERBICIDAL 2-(4,4-DISUBSTITUTED 5-OXO-2-IMIDAZOLIN-2-YL)BENZOIC, NICOTINIC AND QUINOLINE-3-CARBOXYLIC ACIDS, ESTERS AND SALTS AMERICAN CYANAMID COMPANY (US) 1993-03-17 EP disclosed
EP-0205879-A2 Process for the preparation of herbicidal 2-(4,4-disubstituted 5-oxo-2-imidazolin-2-yl)benzoic, nicotinic and quinoline-3-carboxylic acids, esters and salts AMERICAN CYANAMID COMPANY (US) 1986-12-30 EP disclosed
EP-0204209-A2 Imidazo-isoquinoline triones, process for their preparation and agents with a herbicidal activity containing them SCHERING AKTIENGESELLSCHAFT (DE) 1986-12-10 EP disclosed