SCHEMBL9607575

SCHEMBL9607575

Cc1nc(C(=O)NCCN(C)C)ncc1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
TLR9 Q9NR96 2/20 0.42
TLR8 Q9NR97 2/20 0.42
TLR7 Q9NYK1 2/20 0.42
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HPGD P15428 2/20 0.40
MAPK1 P28482 1/20 0.38
ALOX5 P09917 1/20 0.38
LMNA P02545 2/20 0.38
HTR2C P28335 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
AKT3 Q9Y243 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16479775 0.80 TLR9 (0.47) ALDH1A1TLR9TLR8TLR7HTT
SCHEMBL25692411 0.76 AKT3 (0.45) ALDH1A1TLR9TLR8TLR7HTT
SCHEMBL24656058 0.74 CHEK2 (0.46) ALDH1A1HTTSMN1; SMN2HPGDMAPK1
SCHEMBL29990909 0.74 CYP1A2 (0.50) ALDH1A1HTTSMN1; SMN2HPGDMAPK1
SCHEMBL16479768 0.74 TLR9 (0.43) ALDH1A1TLR9TLR8TLR7HTT
SCHEMBL14572014 0.71 ALDH1A1 (0.50) ALDH1A1TLR9TLR8TLR7HTT
SCHEMBL12985976 0.69 NPC1 (0.54) ALDH1A1TLR9TLR8TLR7HTT
SCHEMBL12247423 0.69 HTR2C (0.47) ALDH1A1TLR9TLR8TLR7HTT
SCHEMBL30865637 0.68 MAPK1 (0.41) ALDH1A1TLR9TLR8TLR7HTT
SCHEMBL24810236 0.68 MAPK1 (0.41) ALDH1A1TLR9TLR8TLR7HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071519-A1 BENZOXAZEPINES AS INHIBITORS OF P13K/MTOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-31 WO disclosed