SCHEMBL9608092

SCHEMBL9608092

N#Cc1cccc(Oc2nc(C#CCCNc3ncnc4ccccc34)cs2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.44
CCNC P24863 2/20 0.42
CDK8 P49336 2/20 0.42
CDKN1A P38936 1/20 0.41
CDK19 Q9BWU1 1/20 0.41
CYP1A2 P05177 8/20 0.39
CYP3A4 P08684 7/20 0.39
CLK4 Q9HAZ1 7/20 0.39
LMNA P02545 7/20 0.39
USP2 O75604 6/20 0.39
HSD17B10 Q99714 6/20 0.39
CYP2D6 P10635 5/20 0.39
TSHR P16473 5/20 0.39
ALDH1A1 P00352 5/20 0.39
CYP2C9 P11712 5/20 0.39
MAPK1 P28482 5/20 0.39
HIF1A Q16665 3/20 0.39
TP53 P04637 3/20 0.39
RECQL P46063 2/20 0.39
CYP2C19 P33261 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9608093 0.91 ABCG2 (0.43) ABCG2CCNCCDK8CDKN1ACDK19
SCHEMBL8506086 0.88 EGFR (0.45) ABCG2CLK4LMNATSHRMAPK1
SCHEMBL9608087 0.88 CLK4 (0.45) ABCG2CDK8CYP1A2CYP3A4CLK4
SCHEMBL9608094 0.88 EGFR (0.41) ABCG2CDK8CLK4LMNAMAPK1
SCHEMBL9608089 0.86 EGFR (0.43) ABCG2LMNATSHRMAPK1LDHA
SCHEMBL9609180 0.84 CCNC (0.49) ABCG2CCNCCDK8CDKN1ACDK19
SCHEMBL8516540 0.83 LDHA (0.40) ABCG2CCNCCDK8CDKN1ACDK19
SCHEMBL8504439 0.83 LDHA (0.41) LMNATSHRMAPK1LDHAEGFR
SCHEMBL9608088 0.83 EGFR (0.50) ABCG2CDK8CLK4LMNAALDH1A1
SCHEMBL9608090 0.81 LDHA (0.39) ABCG2CYP1A2CYP3A4CLK4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9089139-B2 Agri-horticultural pest control compositions comprising 4-(3-butynyl)aminopyrimidine derivatives SDS BIOTECH K. K. (JP) 2015-07-28 US disclosed
US-9089139-B2 Agri-horticultural pest control compositions comprising 4-(3-butynyl)aminopyrimidine derivatives SDS BIOTECH K. K. (JP) 2015-07-28 US disclosed
US-8586505-B2 4-(3-butynyl)aminopyrimidine derivatives as pest control agents for agricultural and horticultural use SDS BIOTECH K. K. (JP) 2013-11-19 US disclosed
US-20130296271-A1 Agri-Horticultural Pest Control Compositions Comprising 4-(3-Butynyl)Aminopyrimidine Derivatives SDS BIOTECH K.K. (JP) 2013-11-07 US disclosed
US-20130296271-A1 Agri-Horticultural Pest Control Compositions Comprising 4-(3-Butynyl)Aminopyrimidine Derivatives SDS BIOTECH K.K. (JP) 2013-11-07 US disclosed
US-20120136150-A1 4-(3-Butynyl)Aminopyrimidine Derivatives as Pest Control Agents for Agricultural and Horticultural Use SDS BIOTECH K.K. (JP) 2012-05-31 US disclosed
WO-2011007839-A1 4-(3-BUTYNYL)AMINOPYRIMIDINE DERIVATIVES AS PEST CONTROL AGENTS FOR AGRICULTURAL AND HORTICULTURAL USE 株式会社エス・ディー・エス バイオテック (JP) 2011-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130296271-A1 Agri-Horticultural Pest Control Compositions Comprising 4-(3-Butynyl)Aminopyrimidine Derivatives HCN1, HCN2, HCN3 ABCG2 1188/4885CCNC 2339/4885CDK8 1404/4885
US-20120136150-A1 4-(3-Butynyl)Aminopyrimidine Derivatives as Pest Control Agents for Agricultural and Horticultural Use CBR3, CBR1, HRH2 ABCG2 3012/4885CCNC 2016/4885CDK8 1131/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.