SCHEMBL9612059

SCHEMBL9612059

CNS(=O)(=O)Cc1cccc(NO)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
MMP1 P03956 1/20 0.44
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
MMP13 P45452 1/20 0.44
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTR6 P50406 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA1A P35348 1/20 0.38
HPGD P15428 1/20 0.38
ALKBH5 Q6P6C2 1/20 0.37
IKBKB O14920 1/20 0.37
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11090677 0.83 NEK2 (0.42) CA1CA2MMP1MMP2MMP9
SCHEMBL9612056 0.83 ALDH1A1 (0.43) CA1CA2MMP1MMP2MMP9
SCHEMBL9612063 0.83 ALDH1A1 (0.41) CA1CA2MMP1MMP2MMP9
SCHEMBL9612055 0.79 CA1 (0.52) CA1CA2MMP1MMP2MMP9
SCHEMBL30680228 0.79 CYP1A2 (0.46) CA1CA2MMP1MMP2MMP9
SCHEMBL26659340 0.79 CYP1A2 (0.46) CA1CA2MMP1MMP2MMP9
SCHEMBL10154047 0.77 ACLY (0.49) ALDH1A1HPGDNR3C1
SCHEMBL2991205 0.76 CA1 (0.46) CA1CA2MMP1MMP2MMP9
SCHEMBL5323045 0.76 TAAR1 (0.51)
SCHEMBL2640501 0.76 HTR6 (0.44) CA1CA2MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137166-B1 4, 6-DISUBSTITUTED AMINOPYRIMIDINE DERIVATIVES AS INHIBITORS OF PROTEIN KINASES INGENIUM PHARMACEUTICALS GMBH (DE) 2012-05-30 EP disclosed