SCHEMBL9613341

SCHEMBL9613341

CC(C)c1ccc(-c2nc(C(=O)O)cs2)cc1

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.69
PTPN1 P18031 3/20 0.54
HPGDS O60760 2/20 0.51
RAB9A P51151 2/20 0.51
GAA P10253 1/20 0.51
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADRB3 P13945 1/20 0.49
NPC1 O15118 1/20 0.49
POLB P06746 1/20 0.49
KDM4E B2RXH2 1/20 0.49
PLA2G10 O15496 1/20 0.48
ACHE P22303 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13757164 0.88 ALDH1A1 (0.53) ALDH1A1PTPN1HPGDSRAB9AGAA
SCHEMBL12894475 0.86 ALDH1A1 (0.51) ALDH1A1HPGDSRAB9AGAANPC1
SCHEMBL12925917 0.84 HSD17B1 (0.49) ALDH1A1PTPN1HPGDSRAB9AGAA
SCHEMBL2638322 0.82 ALDH1A1 (0.55) ALDH1A1PTPN1HPGDSADRB2ADRB1
SCHEMBL3412110 0.82 ALDH1A1 (0.71) ALDH1A1PTPN1HPGDSRAB9AGAA
SCHEMBL10037306 0.82 ALDH1A1 (0.71) ALDH1A1PTPN1HPGDSRAB9AGAA
SCHEMBL3098211 0.82 ALDH1A1 (1.00) ALDH1A1PTPN1HPGDSRAB9AGAA
Hydrochloric Acid SCHEMBL6821165 0.81 ALDH1A1 (0.69) ALDH1A1PTPN1HPGDSRAB9AGAA
Hydrochloric Acid SCHEMBL6822031 0.81 ALDH1A1 (0.97) ALDH1A1PTPN1HPGDSRAB9AGAA
SCHEMBL29911269 0.80 RAB9A (0.66) ALDH1A1RAB9AGAANPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727797-B1 PROCESS FOR CROSS COUPLING INDOLES BOEHRINGER INGELHEIM PHARMA (US) 2012-05-30 EP disclosed
US-7893084-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM CANADA LTD. (CA) 2011-02-22 US disclosed
US-7893084-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM CANADA LTD. (CA) 2011-02-22 US disclosed
US-7576079-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2009-08-18 US disclosed
US-20090087409-A1 Viral Polymerase Inhibitors BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2009-04-02 US disclosed
US-20090087409-A1 Viral Polymerase Inhibitors BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2009-04-02 US disclosed
US-7223785-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-29 US disclosed
US-7223785-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-29 US disclosed
EP-0262873-B1 N-TETRAZOLYL THIAZOLECARBOXAMIDE DERIVATIVES AND THEIR USE SAWAI PHARMACEUTICAL CO., LTD. (JP) 1991-08-21 EP disclosed
US-4879295-A ANTIALLERGENS SAWAI PHARMACEUTICAL CO., LTD. (JP) 1989-11-07 US disclosed
EP-0262873-A1 N-tetrazolyl thiazolecarboxamide derivatives and their use SAWAI PHARMACEUTICAL CO., LTD. (JP) 1988-04-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090087409-A1 Viral Polymerase Inhibitors NR2C2, NR4A1, MED25 ALDH1A1 3616/4885PTPN1 642/4885HPGDS 4641/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.