SCHEMBL9617435

SCHEMBL9617435

CC(C)(C)OC(=O)c1ccc(CCCC2CCNc3nc(N)nc(N)c32)cc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.40
NOS1 P29475 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
MTR Q99707 2/20 0.32
LIPC P11150 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
PTGS1 P23219 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997437 0.92 DHFR (0.44) DHFRNOS1SIRT2SIRT1PTGS1
SCHEMBL8569916 0.84 MTR (0.41) DHFRSIRT2SIRT1MTR
SCHEMBL8997208 0.79 DHFR (0.38) DHFRNOS1SIRT2SIRT1PTGS1
SCHEMBL8562117 0.78 MTR (0.44) DHFRSIRT2SIRT1MTR
SCHEMBL9439499 0.75 DHFR (0.46) DHFRNOS1SIRT2SIRT1
SCHEMBL8997222 0.75 DHFR (0.36) DHFRNOS1SIRT2SIRT1
SCHEMBL9446094 0.74
SCHEMBL8997209 0.72 CYP4A11 (0.43) DHFRNOS1
SCHEMBL9446064 0.69 MTR (0.36) MTR
SCHEMBL9446114 0.69 DHFR (0.46) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4235986-A None JP disclosed
JP-H04235986-A PYRIDOPYRIMIDINE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA CHEM IND LTD 1992-08-25 JP disclosed