SCHEMBL8569916

SCHEMBL8569916

CC(C)(C)OC(=O)c1ccc(CCCC2CCc3nc(N)nc(N)c32)cc1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTR Q99707 7/20 0.41
DHFR P00374 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562117 0.94 MTR (0.44) MTRDHFRSIRT2SIRT1
SCHEMBL9617435 0.84 DHFR (0.40) MTRDHFRSIRT2SIRT1
SCHEMBL9446094 0.83
SCHEMBL8997437 0.82 DHFR (0.44) DHFRSIRT2SIRT1
SCHEMBL8571693 0.82 MTR (0.34) MTRSIRT2SIRT1
SCHEMBL9446064 0.79 MTR (0.36) MTR
SCHEMBL8566937 0.78 MTR (0.44) MTRDHFR
SCHEMBL9001819 0.78 ATIC (0.37) MTRSIRT2SIRT1
SCHEMBL8997208 0.76 DHFR (0.38) DHFRSIRT2SIRT1
SCHEMBL1066004 0.73 DHFR (0.59) MTRDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed