SCHEMBL9620680

SCHEMBL9620680

CCOc1cc2c(cc1OCC)C(=O)CCC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.51
HSD17B1 P14061 1/20 0.47
MEN1 O00255 1/20 0.46
MAPK1 P28482 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MAOA P21397 9/20 0.43
MAOB P27338 9/20 0.43
ABCC4 O15439 1/20 0.43
ABCB11 O95342 1/20 0.43
CHRM2 P08172 1/20 0.43
ADRA2A P08913 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CHRM1 P11229 1/20 0.43
PTGS1 P23219 1/20 0.43
PDE4A P27815 1/20 0.43
SLC6A4 P31645 1/20 0.43
KCNH2 Q12809 1/20 0.43
PRKCI P41743 1/20 0.42
PDE4D Q08499 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3082824 0.89 ACHE (0.54) ACHEHSD17B1KMT2AMAOBABCC4
SCHEMBL9621241 0.87 HSD17B1 (0.45) HSD17B1MEN1MAPK1KMT2ANPSR1
SCHEMBL424613 0.80 HSD17B1 (0.54) ACHEHSD17B1MEN1MAPK1KMT2A
SCHEMBL17043164 0.80 ACHE (0.42) ACHEHSD17B1KMT2AMAOBABCC4
SCHEMBL19573418 0.78 MAOB (0.37) ACHEHSD17B1MEN1MAPK1KMT2A
SCHEMBL1545212 0.77 HSD17B1 (0.46) ACHEHSD17B1MEN1MAPK1KMT2A
SCHEMBL8712272 0.77 HSD17B1 (0.46) ACHEHSD17B1MEN1MAPK1KMT2A
SCHEMBL2912990 0.77 MAPT (0.48) ACHEMAPK1ABCC4ABCB11CHRM2
SCHEMBL3083342 0.77 HSD17B1 (0.46) ACHEHSD17B1MEN1KMT2AMAOA
SCHEMBL30701777 0.77 HTR2A (0.43) ACHEHSD17B1MEN1KMT2AABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284359-B1 1,4-DISUBSTITUTED PIPERAZINE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-01-08 EP disclosed
US-4880809-A HYPOTENSIVE AGENTS, AMIDE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-11-14 US disclosed
CN-88101588-A Preparation 1, the method for 4-disubstituted piperazines compounds 1988-11-23 CN disclosed