SCHEMBL9620754

SCHEMBL9620754

COc1cccc2sc(-c3ccc(C)cc3)nc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.56
CYP3A4 P08684 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
KDM4E B2RXH2 6/20 0.52
MAPT P10636 6/20 0.52
MEN1 O00255 2/20 0.52
GAA P10253 2/20 0.52
KMT2A Q03164 2/20 0.52
RAB9A P51151 6/20 0.48
HPGD P15428 6/20 0.48
SMN1; SMN2 Q16637 5/20 0.48
NPC1 O15118 4/20 0.48
TP53 P04637 4/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
DYRK1A Q13627 1/20 0.48
F2RL3 Q96RI0 2/20 0.47
PKM P14618 1/20 0.47
TNKS O95271 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13806222 0.88 ALDH1A1 (0.56) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL9620827 0.88 KDM4E (0.61) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL143850 0.88 ALDH1A1 (0.59) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL1983852 0.87 CYP3A4 (0.63) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL8014076 0.84 TNF (0.57) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL6937797 0.84 APP (0.57) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL8010166 0.83 ALDH1A1 (0.51) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL9620871 0.83 DYRK1A (0.53) ALDH1A1CYP3A4TDP1KDM4EMAPT
SCHEMBL1223274 0.82 APP (0.44) ALDH1A1KDM4EMAPTGAARAB9A
SCHEMBL12422442 0.81 APP (0.58) ALDH1A1CYP3A4TDP1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306708-B1 NOVEL BENZOTHIAZOLE AND ANTIRHEUMATIC AGENT COMPRISING IT AS AN ACTIVE INGREDIENT KANEBO, LTD. (JP) 1992-01-08 EP disclosed
US-4910211-A Containing a phenyl substituted in position 2 and an ester in position 4 KANEBO LTD. (JP) 1990-03-20 US disclosed
EP-0306708-A1 Novel benzothiazole and antirheumatic agent comprising it as an active ingredient KANEBO, LTD. (JP) 1989-03-15 EP disclosed