SCHEMBL9620941

SCHEMBL9620941

O=C(O)C1CCCc2cc(OCc3ccccc3)c(OCc3ccccc3)cc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
FABP4 P15090 1/20 0.42
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
SGMS2 Q8NHU3 1/20 0.40
S1PR5 Q9H228 1/20 0.40
RXRB P28702 2/20 0.40
RXRA P19793 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.40
PTGER1 P34995 1/20 0.39
AGTR2 P50052 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MCL1 Q07820 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9621341 0.94 CHRNA7 (0.47) AGTR2
SCHEMBL9621233 0.86 NPC1 (0.46)
SCHEMBL9621088 0.81 NPC1 (0.43) FABP4
SCHEMBL9620722 0.78 ACHE (0.48)
SCHEMBL21092400 0.78 MAOB (0.43) MAOAMAOBALDH1A1
SCHEMBL21054283 0.78 MAOB (0.43) MAOAMAOBALDH1A1
SCHEMBL7278343 0.77 MAOA (0.68) MAOAMAOBMRGPRX4
SCHEMBL9620731 0.75 ACHE (0.47)
SCHEMBL7223230 0.74 MAOA (0.58) MAOAMAOBMEN1ALDH1A1KMT2A
SCHEMBL7281372 0.74 CHRNA7 (0.51) MAOBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284359-B1 1,4-DISUBSTITUTED PIPERAZINE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-01-08 EP disclosed
US-4880809-A HYPOTENSIVE AGENTS, AMIDE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-11-14 US disclosed
EP-0284359-A1 1,4-Disubstituted piperazine compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-09-28 EP disclosed