SCHEMBL9621922

SCHEMBL9621922

C=CC(NCc1ccccc1)N1CCCC1=O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 2/20 0.37
SLC1A2 P43004 1/20 0.36
POLB P06746 3/20 0.36
ACP3 P15309 3/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5431412 0.71 CHRM2 (0.47) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL8522922 0.70 SLC6A4 (0.47) SMN1; SMN2KMT2A
SCHEMBL22558182 0.69 SLC1A2 (0.67) SMN1; SMN2LMNAKMT2ASLC1A2HTT
SCHEMBL22558181 0.69 SLC1A2 (0.67) SMN1; SMN2LMNAKMT2ASLC1A2HTT
SCHEMBL30495979 0.69 SLC1A2 (0.67) SMN1; SMN2LMNAKMT2ASLC1A2HTT
SCHEMBL9461581 0.68 LMNA (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL27603655 0.67 L3MBTL1 (0.46) SMN1; SMN2L3MBTL1LMNAKMT2ASLC1A2
N-Benzylmethylamine SCHEMBL29834172 0.67 LMNA (0.53) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11347598 0.67 SLC1A2 (0.50) KMT2ASLC1A2
SCHEMBL18836847 0.67 NPC1 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0136658-B1 -1-BENZYL-AMINOALKYL-PYRROLIDINONES AND THEIR ADDITION SALTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUNDS CONTAINING THEM BOEHRINGER INGELHEIM KG (DE) 1989-04-26 EP claimed
EP-0136658-A2 -1-Benzyl-aminoalkyl-pyrrolidinones and their addition salts, process for their preparation and pharmaceutical compounds containing them BOEHRINGER INGELHEIM KG (DE) 1985-04-10 EP claimed
JP-4261152-A None JP disclosed
JP-H04261152-A NOVEL 1-BENZYL-AMINOALKYL-PYRROLIDINONE COMPOUND AND ITS PRODUCTION BOEHRINGER INGELHEIM KG 1992-09-17 JP disclosed
EP-0266563-B1 USE OF 1-BENZYL-AMINO-ALKYL-PYRROLIDINONES AS ANTIDEPRESSANTS BOEHRINGER INGELHEIM KG (DE) 1992-01-29 EP disclosed
EP-0266563-B1 USE OF 1-BENZYL-AMINO-ALKYL-PYRROLIDINONES AS ANTIDEPRESSANTS BOEHRINGER INGELHEIM KG (DE) 1992-01-29 EP disclosed
US-4954516-A Use of 1-benzyl-aminoalkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1990-09-04 US disclosed
US-4954516-A Use of 1-benzyl-aminoalkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1990-09-04 US disclosed
US-4954516-A Use of 1-benzyl-aminoalkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1990-09-04 US disclosed
US-4912129-A Administering to humans BOEHRINGER INGELHEIM GMBH (DE) 1990-03-27 US disclosed
US-4912129-A Administering to humans BOEHRINGER INGELHEIM GMBH (DE) 1990-03-27 US disclosed
EP-0136658-B1 -1-BENZYL-AMINOALKYL-PYRROLIDINONES AND THEIR ADDITION SALTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUNDS CONTAINING THEM BOEHRINGER INGELHEIM KG (DE) 1989-04-26 EP disclosed
US-4812453-A Use of 1-benzyl-aminoalkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1989-03-14 US disclosed
US-4812453-A Use of 1-benzyl-aminoalkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1989-03-14 US disclosed
US-4812453-A Use of 1-benzyl-aminoalkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1989-03-14 US disclosed
EP-0266563-A2 Use of 1-benzyl-amino-alkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1988-05-11 EP disclosed
EP-0266563-A2 Use of 1-benzyl-amino-alkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1988-05-11 EP disclosed
EP-0266563-A2 Use of 1-benzyl-amino-alkyl-pyrrolidinones as antidepressants BOEHRINGER INGELHEIM KG (DE) 1988-05-11 EP disclosed
EP-0136658-A2 -1-Benzyl-aminoalkyl-pyrrolidinones and their addition salts, process for their preparation and pharmaceutical compounds containing them BOEHRINGER INGELHEIM KG (DE) 1985-04-10 EP disclosed
EP-0136658-A2 -1-Benzyl-aminoalkyl-pyrrolidinones and their addition salts, process for their preparation and pharmaceutical compounds containing them BOEHRINGER INGELHEIM KG (DE) 1985-04-10 EP disclosed