SCHEMBL9622351

SCHEMBL9622351

COC(=O)C(=O)CC(CO[Si](C)(C)C(C)(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 9/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CYP2D6 P10635 1/20 0.35
SYK P43405 1/20 0.35
ATM Q13315 1/20 0.33
AAK1 Q2M2I8 2/20 0.33
CTSS P25774 4/20 0.33
CTSL P07711 1/20 0.33
KMT2A Q03164 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10487514 0.86 SMN1; SMN2 (0.40) CTSKCA1CA2CA7CYP2D6
SCHEMBL7346754 0.85 CA1 (0.38) CTSKCA1CA2CA7CYP2D6
SCHEMBL4520424 0.85 CA1 (0.38) CTSKCA1CA2CA7CYP2D6
SCHEMBL1262397 0.85 CA1 (0.38) CTSKCA1CA2CA7CYP2D6
SCHEMBL1861342 0.82 CA1 (0.40) CTSKCA1CA2CA7CYP2D6
SCHEMBL3227264 0.82 CA1 (0.40) CTSKCA1CA2CA7CYP2D6
SCHEMBL1861340 0.82 CA1 (0.40) CTSKCA1CA2CA7CYP2D6
SCHEMBL28343011 0.81 CTSK (0.43) CTSKCA1CA2CA7CYP2D6
SCHEMBL28343009 0.81 CTSK (0.43) CTSKCA1CA2CA7CYP2D6
SCHEMBL3613413 0.81 CA1 (0.39) CTSKCA1CA2CA7CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4588825-A Intermediates for the synthesis of 4-amino-4,5-dihydro-2-furancarboxylic acid MERRELL DOW PHARMACEUTICALS INC. (US) 1986-05-13 US claimed
EP-0145875-A2 Gamma-aminobutyric acid transaminase inhibitors and processes for their preparation MERRELL DOW PHARMACEUTICALS INC. (US) 1985-06-26 EP claimed
EP-0145875-B1 GAMMA-AMINOBUTYRIC ACID TRANSAMINASE INHIBITORS AND PROCESSES FOR THEIR PREPARATION MERRELL DOW PHARMACEUTICALS INC. (US) 1992-02-19 EP disclosed
US-4824974-A Synthesis for the preparation of 4-amino-4,5-dihydro-2-furancarboxylic acid MERRELL DOW PHARMACEUTICALS INC. (US) 1989-04-25 US disclosed
US-4588825-A Intermediates for the synthesis of 4-amino-4,5-dihydro-2-furancarboxylic acid MERRELL DOW PHARMACEUTICALS INC. (US) 1986-05-13 US disclosed
EP-0145875-A2 Gamma-aminobutyric acid transaminase inhibitors and processes for their preparation MERRELL DOW PHARMACEUTICALS INC. (US) 1985-06-26 EP disclosed