SCHEMBL3227264

SCHEMBL3227264

CC(C)(C)OC(=O)N[C@H](CO)CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
ATM Q13315 1/20 0.36
CTSK P43235 6/20 0.36
CYP2D6 P10635 1/20 0.36
AAK1 Q2M2I8 4/20 0.35
KMT2A Q03164 1/20 0.35
CTSS P25774 2/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1861340 1.00 CA1 (0.40) CA1CA2CA7ATMCTSK
SCHEMBL1861342 1.00 CA1 (0.40) CA1CA2CA7ATMCTSK
SCHEMBL31695224 0.88 CA1 (0.35) CA1CA2CA7ATMCTSK
SCHEMBL30732579 0.88 CA1 (0.35) CA1CA2CA7ATMCTSK
SCHEMBL3613413 0.87 CA1 (0.39) CA1CA2CA7ATMCTSK
SCHEMBL3613415 0.87 CA1 (0.39) CA1CA2CA7ATMCTSK
SCHEMBL213446 0.86 TDP1 (0.40) CA1CA2CA7ATMCTSK
SCHEMBL211028 0.86 CA1 (0.36) CA1CA2CA7ATMCTSK
SCHEMBL213445 0.86 TDP1 (0.40) CA1CA2CA7ATMCTSK
SCHEMBL211029 0.86 CA1 (0.36) CA1CA2CA7ATMCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3413922-B1 IMPROVED SULFAMIDE LINKERS FOR USE IN BIOCONJUGATES SYNAFFIX BV (NL) 2025-12-10 EP disclosed
US-20250353848-A1 HETEROCYCLIC PAD4 INHIBITORS CELGENE CORPORATION 2025-11-20 US disclosed
US-20250346592-A1 HETEROCYCLIC PAD4 INHIBITORS CELGENE CORPORATION 2025-11-13 US disclosed
US-12384797-B2 Thioeno[3,2-b] pyridin-7-amine compounds for treating familial dysautonomia PTC THERAPEUTICS, INC. (US) 2025-08-12 US disclosed
WO-2025137639-A1 MIXED SEROTONIN RECEPTOR BINDERS FOR TREATMENT OF PSYCHOTIC DISORDERS DELIX THERAPEUTICS, INC. (US) 2025-06-26 WO disclosed
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME MONTE ROSA THERAPEUTICS AG (CH) 2025-05-29 US disclosed
EP-4540240-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME Monte Rosa Therapeutics AG (CH) 2025-04-23 EP disclosed
EP-4531849-A1 HETEROCYCLIC PAD4 INHIBITORS CELGENE CORPORATION (US) 2025-04-09 EP disclosed
US-11957763-B2 Sulfamide linkers for use in bioconjugates SYNAFFIX B.V. (NL) 2024-04-16 US disclosed
WO-2023244815-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME MONTE ROSA THERAPEUTICS, INC. (US) 2023-12-21 WO disclosed
US-20080318945-A1 Novel Compounds CASILLAS LINDA N 2008-12-25 US disclosed
US-20080318945-A1 Novel Compounds CASILLAS LINDA N 2008-12-25 US disclosed
US-20080293712-A1 Benzo[C][2,7]Naphtyridine Derivatives, Methods of Making Thereof and Methods of Use Thereof WYETH (US) 2008-11-27 US disclosed
US-20070225267-A1 3-(2-Acylamino-1-Hydroxyethyl)-Morpholine Derivatives and Their Use as Bace Inhibitors ELI LILLY AND COMPANY 2007-09-27 US disclosed
US-20070185152-A1 Inhibitors of akt activity SMITHKLINE BEECHAM CORPORATION 2007-08-09 US disclosed
WO-2007070865-A2 PIPERAZINE COMPOUNDS AS AGONISTS OF TRPV4 CHANNEL RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2007-06-21 WO disclosed
WO-2006034093-A2 3- (2-ACYLAMINO-1-HYDROXYETHYL)- MORPHOLINE DERIVATIVES AND THEIR USE AS BACE INHIBITORS ELLI LILLY AND COMPANY (US) 2006-03-30 WO disclosed
US-6831175-B2 Such as N,N-dimethyl-N-(2-((5-((E)-2-pyridin-4-ylvinyl) pyridin-3-yl)oxy)ethyl)amine ABBOTT LABORATORIES 2004-12-14 US disclosed
US-20030199511-A1 Kinase inhibitors ABBVIE INC. 2003-10-23 US disclosed
US-20030187026-A1 Kinase inhibitors ABBOTT LABORATORIES 2003-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250353848-A1 HETEROCYCLIC PAD4 INHIBITORS PADI4, PADI1, PADI6 CA1 3667/4885CA2 4042/4885CA7 2790/4885
US-20080318945-A1 Novel Compounds TRPV4, TRPV1, TRPV3 CA1 3946/4885CA2 520/4885CA7 2877/4885
US-11957763-B2 Sulfamide linkers for use in bioconjugates CD22, SPG11, SP1 CA1 934/4885CA2 2442/4885CA7 1047/4885
US-20030187026-A1 Kinase inhibitors MAP3K20, MAP3K19, MAP3K1 CA1 3197/4885CA2 2667/4885CA7 2522/4885
US-20070185152-A1 Inhibitors of akt activity AKT1, AKT1S1, AKT2 CA1 3648/4885CA2 3883/4885CA7 3427/4885
US-20030199511-A1 Kinase inhibitors MAP3K20, MAP3K19, MAP3K1 CA1 3197/4885CA2 2667/4885CA7 2522/4885
US-20070225267-A1 3-(2-Acylamino-1-Hydroxyethyl)-Morpholine Derivatives and Their Use as Bace Inhibitors BACE1, BACE2, APP CA1 1464/4885CA2 2660/4885CA7 1442/4885
US-12384797-B2 Thioeno[3,2-b] pyridin-7-amine compounds for treating familial dysautonomia SF3B5, SF3B2, SF3B1 CA1 4838/4885CA2 4657/4885CA7 4739/4885
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME PSMA1, CSNK1G1, CSNK1A1 CA1 855/4885CA2 1677/4885CA7 1209/4885
US-20250346592-A1 HETEROCYCLIC PAD4 INHIBITORS PADI4, PADI6, PADI2 CA1 2957/4885CA2 3840/4885CA7 3010/4885
US-20080293712-A1 Benzo[C][2,7]Naphtyridine Derivatives, Methods of Making Thereof and Methods of Use Thereof PDPK1, PDK2, PDK3 CA1 3315/4885CA2 1620/4885CA7 926/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.