SCHEMBL9622953

SCHEMBL9622953

CC(=O)Nc1ccc(C(=O)NCC2(O)CN3CCC2CC3)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.45
NR1H4 Q96RI1 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
ALDH1A1 P00352 4/20 0.43
NFKB1 P19838 1/20 0.43
KCNH2 Q12809 1/20 0.43
HTT P42858 2/20 0.43
NAMPT P43490 2/20 0.43
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
THRB P10828 1/20 0.43
BLM P54132 1/20 0.43
ATM Q13315 1/20 0.43
MAPK14 Q16539 1/20 0.42
TP53 P04637 1/20 0.42
HIF1A Q16665 1/20 0.42
CACNA1B Q00975 1/20 0.42
APBA1 Q02410 1/20 0.42
TSHR P16473 1/20 0.41
MMP13 P45452 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9622879 0.84 SMN1; SMN2 (0.49) EPHX2NR1H4SMN1; SMN2ALDH1A1HTT
Water SCHEMBL9623050 0.83 SMN1; SMN2 (0.48) EPHX2NR1H4SMN1; SMN2ALDH1A1HTT
Water SCHEMBL9623052 0.83 SMN1; SMN2 (0.48) EPHX2NR1H4SMN1; SMN2ALDH1A1HTT
SCHEMBL9623214 0.83 NSD2 (0.44) EPHX2POLBHIF1AMMP13KDM4E
SCHEMBL8772585 0.77 KMT2A (0.49) SMN1; SMN2ALDH1A1HTT
SCHEMBL9622615 0.74 SIGMAR1 (0.45) MMP13MMP2
SCHEMBL6257293 0.71 MAPK14 (0.70) EPHX2NR1H4SMN1; SMN2ALDH1A1NFKB1
SCHEMBL8772657 0.70 MMP13 (0.62) MMP13MMP2
SCHEMBL9622442 0.69 BCHE (0.52) ALDH1A1
SCHEMBL5508324 0.69 ALDH1A1 (0.70) EPHX2NR1H4SMN1; SMN2ALDH1A1NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5137895-A Antiemetic, anxiolytic, gastric emptying and serotonin modulating activity A. H. ROBINS COMPANY, INCORPORATED (US) 1992-08-11 US disclosed